Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50006193
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045906(3-Oxo-hexadecanoic acid (2,6-diisopropyl-phenyl)-a...)
Affinity DataIC50: 6nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045911(3-Oxo-pentadecanoic acid (2,6-diisopropyl-phenyl)-...)
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045915(N-(2,6-Diisopropyl-phenyl)-3-oxo-3-(1-phenyl-cyclo...)
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045919(7-Dodecyl-2-oxo-azepane-3-carboxylic acid (2,6-dii...)
Affinity DataIC50: 22nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045902(3-Oxo-heptadecanoic acid (2,6-diisopropyl-phenyl)-...)
Affinity DataIC50: 24nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045914(N-(2,6-Diisopropyl-phenyl)-3-oxo-4,4-diphenyl-buty...)
Affinity DataIC50: 35nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045909(3-Oxo-5,5-diphenyl-pentanoic acid (2,6-diisopropyl...)
Affinity DataIC50: 44nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045907(5-Dodecyl-2-oxo-pyrrolidine-3-carboxylic acid (2,6...)
Affinity DataIC50: 53nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045910(3-Oxo-13-(tetrahydro-pyran-2-yloxy)-tridecanoic ac...)
Affinity DataIC50: 57nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045916(3-Oxo-tridecanoic acid (2,6-diisopropyl-phenyl)-am...)
Affinity DataIC50: 60nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045918(3-Oxo-tetradecanoic acid (2,6-diisopropyl-phenyl)-...)
Affinity DataIC50: 69nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045908(3-Oxo-dodecanoic acid (2,6-diisopropyl-phenyl)-ami...)
Affinity DataIC50: 97nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045898(3-Oxo-tetradecanoic acid (2,4,6-trimethoxy-phenyl)...)
Affinity DataIC50: 150nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045913(3-Hydroxyimino-5,5-diphenyl-pentanoic acid (2,6-di...)
Affinity DataIC50: 210nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045904(13-Hydroxy-3-oxo-tridecanoic acid (2,6-diisopropyl...)
Affinity DataIC50: 230nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045899(5-Heptyl-2-oxo-tetrahydro-furan-3-carboxylic acid ...)
Affinity DataIC50: 260nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045905(6-Heptyl-2-oxo-tetrahydro-pyran-3-carboxylic acid ...)
Affinity DataIC50: 340nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045897(2,2-Dimethyl-3-oxo-tetradecanoic acid (2,4,6-trime...)
Affinity DataIC50: 370nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045903(6-Hexyl-2-oxo-tetrahydro-pyran-3-carboxylic acid (...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045901(N-(2,6-Diisopropyl-phenyl)-3-oxo-3-phenyl-propiona...)
Affinity DataIC50: 810nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045912(2,2-Dimethyl-3-oxo-tetradecanoic acid methyl-(2,4,...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045917(2,2-Dimethyl-3-oxo-tetradecanoic acid (2,6-diisopr...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045900(3-Hydroxy-5,5-diphenyl-pentanoic acid (2,6-diisopr...)
Affinity DataIC50: 3.50E+3nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase in intestinal microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed