Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 5026
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi:  1.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi:  1.58nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi:  1.99nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi:  12.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi:  50.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi:  398nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi:  398nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi:  501nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi:  794nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi:  1.26E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi:  1.26E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi:  1.26E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi:  2.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi:  2.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi:  2.51E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi:  5.01E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi:  6.31E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Pig)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Pig)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rhesus macaque)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rhesus macaque)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84951(CAS_133075 | NSC_133075 | RS 67506)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed