Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50006458
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataIC50: 6nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049365(1-benzyl-4-(2-(bis(4-fluorophenyl)methoxy)ethyl)pi...)
Affinity DataIC50: 9.70nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049360(4-(2-Benzhydryloxy-ethyl)-1-phenethyl-piperidine |...)
Affinity DataIC50: 10.6nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049359(4-(2-Benzhydryloxy-ethyl)-1-(3-phenyl-propyl)-pipe...)
Affinity DataIC50: 12nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049371(4-[Bis-(4-fluoro-phenyl)-methoxymethyl]-1-(3-pheny...)
Affinity DataIC50: 13nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049364(4-[Bis-(4-fluoro-phenyl)-methoxymethyl]-1-phenethy...)
Affinity DataIC50: 13.5nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049369(4-Benzhydryloxymethyl-1-(3-phenyl-propyl)-piperidi...)
Affinity DataIC50: 14.5nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049362(4-(2-Benzhydryloxy-ethyl)-1-benzyl-piperidine | CH...)
Affinity DataIC50: 15.2nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049363(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(3-p...)
Affinity DataIC50: 16.7nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049357(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-phen...)
Affinity DataIC50: 19.9nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049357(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-phen...)
Affinity DataIC50: 31.9nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049363(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(3-p...)
Affinity DataIC50: 55nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049369(4-Benzhydryloxymethyl-1-(3-phenyl-propyl)-piperidi...)
Affinity DataIC50: 58nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049372(4-{2-[Bis-(4-chloro-phenyl)-methoxy]-ethyl}-1-(3-p...)
Affinity DataIC50: 65nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataIC50: 82nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049360(4-(2-Benzhydryloxy-ethyl)-1-phenethyl-piperidine |...)
Affinity DataIC50: 102nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049358(4-Benzhydryloxymethyl-1-phenethyl-piperidine | CHE...)
Affinity DataIC50: 108nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049371(4-[Bis-(4-fluoro-phenyl)-methoxymethyl]-1-(3-pheny...)
Affinity DataIC50: 112nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049367(4-{2-[Bis-(4-chloro-phenyl)-methoxy]-ethyl}-1-phen...)
Affinity DataIC50: 115nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049373(1-Benzyl-4-[bis-(4-fluoro-phenyl)-methoxymethyl]-p...)
Affinity DataIC50: 126nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049368(4-{2-[Bis-(4-bromo-phenyl)-methoxy]-ethyl}-1-(3-ph...)
Affinity DataIC50: 159nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049365(1-benzyl-4-(2-(bis(4-fluorophenyl)methoxy)ethyl)pi...)
Affinity DataIC50: 198nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049372(4-{2-[Bis-(4-chloro-phenyl)-methoxy]-ethyl}-1-(3-p...)
Affinity DataIC50: 224nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049359(4-(2-Benzhydryloxy-ethyl)-1-(3-phenyl-propyl)-pipe...)
Affinity DataIC50: 232nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049364(4-[Bis-(4-fluoro-phenyl)-methoxymethyl]-1-phenethy...)
Affinity DataIC50: 237nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049361(4-{2-[Bis-(4-methoxy-phenyl)-methoxy]-ethyl}-1-(3-...)
Affinity DataIC50: 255nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049374(4-(2-Di-p-tolylmethoxy-ethyl)-1-phenethyl-piperidi...)
Affinity DataIC50: 311nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049361(4-{2-[Bis-(4-methoxy-phenyl)-methoxy]-ethyl}-1-(3-...)
Affinity DataIC50: 340nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049366(4-{2-[Bis-(4-bromo-phenyl)-methoxy]-ethyl}-1-phene...)
Affinity DataIC50: 382nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049367(4-{2-[Bis-(4-chloro-phenyl)-methoxy]-ethyl}-1-phen...)
Affinity DataIC50: 414nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049358(4-Benzhydryloxymethyl-1-phenethyl-piperidine | CHE...)
Affinity DataIC50: 456nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049370(4-Benzhydryloxymethyl-1-benzyl-piperidine | CHEMBL...)
Affinity DataIC50: 544nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049366(4-{2-[Bis-(4-bromo-phenyl)-methoxy]-ethyl}-1-phene...)
Affinity DataIC50: 638nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50049370(4-Benzhydryloxymethyl-1-benzyl-piperidine | CHEMBL...)
Affinity DataIC50: 702nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]CFT displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049362(4-(2-Benzhydryloxy-ethyl)-1-benzyl-piperidine | CH...)
Affinity DataIC50: 743nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049373(1-Benzyl-4-[bis-(4-fluoro-phenyl)-methoxymethyl]-p...)
Affinity DataIC50: 761nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049368(4-{2-[Bis-(4-bromo-phenyl)-methoxy]-ethyl}-1-(3-ph...)
Affinity DataIC50: 835nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049374(4-(2-Di-p-tolylmethoxy-ethyl)-1-phenethyl-piperidi...)
Affinity DataIC50: 888nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]citalopram displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed