Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50003429
TargetD(4) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470855(CHEMBL60708)
Affinity DataKi:  4nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470850(CHEMBL59326)
Affinity DataKi:  5nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470854(CHEMBL433255)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50203469(3-Methoxy-naphthalene-2-carboxylic acid (1-benzyl-...)
Affinity DataKi:  20nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470852(CHEMBL57019)
Affinity DataKi:  20nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470857(CHEMBL299479)
Affinity DataKi:  25nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470849(CHEMBL59075)
Affinity DataKi:  25nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470851(CHEMBL57407)
Affinity DataKi:  32nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470856(CHEMBL292186)
Affinity DataKi:  32nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470855(CHEMBL60708)
Affinity DataKi:  40nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50203469(3-Methoxy-naphthalene-2-carboxylic acid (1-benzyl-...)
Affinity DataKi:  126nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470853(CHEMBL61090)
Affinity DataKi:  200nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470856(CHEMBL292186)
Affinity DataKi:  398nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470851(CHEMBL57407)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470853(CHEMBL61090)
Affinity DataKi:  1.26E+3nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470849(CHEMBL59075)
Affinity DataKi:  1.59E+3nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470857(CHEMBL299479)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470850(CHEMBL59326)
Affinity DataKi:  3.16E+3nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470854(CHEMBL433255)
Affinity DataKi:  7.94E+3nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470852(CHEMBL57019)
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed