Compile Data Set for Download or QSAR
Report error Found 121 Enz. Inhib. hit(s) with all data for entry = 50006566
TargetMetabotropic glutamate receptor 2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50076393((1S,2S,3R)-2-((S)-Amino-carboxy-methyl)-3-phenyl-c...)
Affinity DataIC50: 8.00E+3nMAssay Description:Concentration required for the half-maximal inhibition of cAMP hydrolysis in BHK cells expressing mGluR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407819(CHEMBL2115152)
Affinity DataKi:  4.40E+4nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50030627(CHEMBL299683 | MCPG | (R,S)-alpha-Methyl-4-carboxy...)
Affinity DataKi:  5.00E+4nMAssay Description:Binding affinity towards mGluR1a was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50076393((1S,2S,3R)-2-((S)-Amino-carboxy-methyl)-3-phenyl-c...)
Affinity DataKi:  5.00E+4nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50030627(CHEMBL299683 | MCPG | (R,S)-alpha-Methyl-4-carboxy...)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonistic activity against mGluR2 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407823(CHEMBL2114116)
Affinity DataKi:  6.00E+4nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407827(CHEMBL2115160)
Affinity DataEC50:  1.22E+5nMAssay Description:Effective concentration forskolin-stimulated cAMP formation in BHK cells expressing mGluR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407827(CHEMBL2115160)
Affinity DataKi:  1.35E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407819(CHEMBL2115152)
Affinity DataIC50: 1.40E+5nMAssay Description:Concentration required for the half-maximal inhibition of PI hydrolysis in BHK cells expressing mGluR1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50076393((1S,2S,3R)-2-((S)-Amino-carboxy-methyl)-3-phenyl-c...)
Affinity DataEC50:  1.56E+5nMAssay Description:Effective concentration of compound against forskolin-stimulated cAMP formation in BHK cells expressing mGluR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407824(CHEMBL2114115)
Affinity DataKi:  2.05E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407822(CHEMBL2114112)
Affinity DataKi:  2.60E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407825(CHEMBL2114110)
Affinity DataKi: >2.70E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407830(CHEMBL2115157)
Affinity DataKi: >2.70E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407829(CHEMBL2115153)
Affinity DataKi: >2.70E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407820(CHEMBL2115159)
Affinity DataKi: >2.70E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407821(CHEMBL2115151)
Affinity DataKi: >2.70E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407828(CHEMBL2114106)
Affinity DataKi: >2.70E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50076393((1S,2S,3R)-2-((S)-Amino-carboxy-methyl)-3-phenyl-c...)
Affinity DataKi: >2.70E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407826(CHEMBL2114105)
Affinity DataKi: >2.70E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407825(CHEMBL2114110)
Affinity DataKi: >2.70E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407818(CHEMBL2114109)
Affinity DataKi: >2.70E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407831(CHEMBL2115156)
Affinity DataKi: >2.70E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407819(CHEMBL2115152)
Affinity DataKi: >2.80E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407822(CHEMBL2114112)
Affinity DataKi: >2.80E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407820(CHEMBL2115159)
Affinity DataKi: >2.80E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407824(CHEMBL2114115)
Affinity DataKi: >2.80E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407828(CHEMBL2114106)
Affinity DataKi: >2.80E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407827(CHEMBL2115160)
Affinity DataKi: >2.80E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407823(CHEMBL2114116)
Affinity DataKi: >2.80E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407825(CHEMBL2114110)
Affinity DataKi: >2.80E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407826(CHEMBL2114105)
Affinity DataKi: >2.80E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407818(CHEMBL2114109)
Affinity DataKi: >2.80E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407830(CHEMBL2115157)
Affinity DataKi: >2.80E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407829(CHEMBL2115153)
Affinity DataKi: >2.80E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407831(CHEMBL2115156)
Affinity DataKi: >2.80E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407821(CHEMBL2115151)
Affinity DataKi: >2.80E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407818(CHEMBL2114109)
Affinity DataEC50: >3.00E+5nMAssay Description:Effective concentration forskolin-stimulated cAMP formation in BHK cells expressing mGluR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407824(CHEMBL2114115)
Affinity DataEC50: >3.00E+5nMAssay Description:Effective concentration against forskolin-stimulated cAMP formation in BHK cells expressing mGluR4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407819(CHEMBL2115152)
Affinity DataEC50: >3.00E+5nMAssay Description:Effective concentration against forskolin-stimulated cAMP formation in BHK cells expressing mGluR4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407827(CHEMBL2115160)
Affinity DataEC50: >3.00E+5nMAssay Description:Concentration required for the half-maximal inhibition of cAMP formation in BHK cells expressing mGluR4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407818(CHEMBL2114109)
Affinity DataEC50: >3.00E+5nMAssay Description:Effective concentration against forskolin-stimulated cAMP formation in BHK cells expressing mGluR4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407827(CHEMBL2115160)
Affinity DataEC50: >3.00E+5nMAssay Description:Concentration required for the half-maximal inhibition of cAMP formation in BHK cells expressing mGluR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407822(CHEMBL2114112)
Affinity DataEC50: >3.00E+5nMAssay Description:Effective concentration forskolin-stimulated cAMP formation in BHK cells expressing mGluR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407830(CHEMBL2115157)
Affinity DataIC50: 3.00E+5nMAssay Description:Concentration required for the half-maximal inhibition of cAMP hydrolysis in BHK cells expressing mGluR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407831(CHEMBL2115156)
Affinity DataIC50: 3.00E+5nMAssay Description:Concentration required for the half-maximal inhibition of PI hydrolysis in BHK cells expressing mGluR1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407831(CHEMBL2115156)
Affinity DataIC50: 3.00E+5nMAssay Description:Concentration required for the half-maximal inhibition of cAMP hydrolysis in BHK cells expressing mGluR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407821(CHEMBL2115151)
Affinity DataIC50: 3.00E+5nMAssay Description:Concentration required for the half-maximal inhibition of cAMP formation in BHK cells expressing mGluR2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407820(CHEMBL2115159)
Affinity DataEC50: >3.00E+5nMAssay Description:Effective concentration against forskolin-stimulated cAMP formation in BHK cells expressing mGluR4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50407823(CHEMBL2114116)
Affinity DataEC50: >3.00E+5nMAssay Description:Effective concentration against forskolin-stimulated cAMP formation in BHK cells expressing mGluR4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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