Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50042210
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1283(3-{[1,3-benzoxazol-2-yl)-methyl]amino}-5-ethyl-6-m...)
Affinity DataIC50: 209nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1284(CHEMBL316785 | Pyridinone deriv. 8 | 3-[(1-benzofu...)
Affinity DataIC50: 331nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1286(5-ethyl-6-methyl-3-[(quinolin-3-ylmethyl)amino]-1,...)
Affinity DataIC50: 339nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1287(3-[(1,3-benzothiazol-2-ylmethyl)amino]-5-ethyl-6-m...)
Affinity DataIC50: 347nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1288(Pyridinone deriv. 10 | 5-ethyl-6-methyl-3-[(naphth...)
Affinity DataIC50: 457nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1289(3-[(1-benzothiophen-2-ylmethyl)amino]-5-ethyl-6-me...)
Affinity DataIC50: 501nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1290(CHEMBL123639 | 5-ethyl-6-methyl-3-[(quinolin-2-ylm...)
Affinity DataIC50: 525nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1293(CHEMBL125873 | 5-ethyl-6-methyl-3-[(naphthalen-1-y...)
Affinity DataIC50: 2.09E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1297(5-ethyl-3-[(1H-indol-2-ylmethyl)amino]-6-methyl-1,...)
Affinity DataIC50: 4.37E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1298(CHEMBL86064 | 2-pyridinone deriv. 28 | 3-(benzylam...)
Affinity DataIC50: 5.37E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1299(CHEMBL98394 | 3-[(1H-1,3-benzodiazol-2-ylmethyl)am...)
Affinity DataIC50: 7.59E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1302(CHEMBL339138 | 5-ethyl-6-methyl-3-[(pyridin-2-ylme...)
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1303(CHEMBL340255 | 5-ethyl-3-[(1H-indol-3-ylmethyl)ami...)
Affinity DataIC50: 2.24E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1304(5-ethyl-3-[(furan-2-ylmethyl)amino]-6-methyl-1,2-d...)
Affinity DataIC50: 2.88E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1305(CHEMBL123735 | 5-ethyl-3-({furo[3,2-c]pyridin-2-yl...)
Affinity DataIC50: 3.24E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1306(5-ethyl-3-({furo[2,3-c]pyridin-2-ylmethyl}amino)-6...)
Affinity DataIC50: 1.05E+5nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1307(5-ethyl-3-[(furan-3-ylmethyl)amino]-6-methyl-1,2-d...)
Affinity DataIC50: 1.45E+5nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Organon Research and Development Group

Curated by ChEMBL
LigandPNGBDBM1308(5-ethyl-6-methyl-3-[(pyridin-3-ylmethyl)amino]-1,2...)
Affinity DataIC50: 3.02E+5nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed