Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 5058
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22541(VUF 9153 | N''-[(4-chlorophenyl)methyl]{[3-(1H-imi...)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM85023(GR-168320 | GR 168320)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM85023(GR-168320 | GR 168320)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22541(VUF 9153 | N''-[(4-chlorophenyl)methyl]{[3-(1H-imi...)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22530(N(alpha)-Methylhistamine | [2-(1H-imidazol-5-yl)et...)
Affinity DataKi:  0.390nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22904(CHEMBL268229 | Alpha-Methylhistane-R | (2R)-1-(1H-...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22904(CHEMBL268229 | Alpha-Methylhistane-R | (2R)-1-(1H-...)
Affinity DataKi:  1.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22530(N(alpha)-Methylhistamine | [2-(1H-imidazol-5-yl)et...)
Affinity DataKi:  1.99nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  1.99nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM7966([3H]histamine | 2-(1H-imidazol-4-yl)ethan-1-amine ...)
Affinity DataKi:  2.51nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22904(CHEMBL268229 | Alpha-Methylhistane-R | (2R)-1-(1H-...)
Affinity DataKi:  3.98nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  3.98nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22530(N(alpha)-Methylhistamine | [2-(1H-imidazol-5-yl)et...)
Affinity DataKi:  5.01nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM7966([3H]histamine | 2-(1H-imidazol-4-yl)ethan-1-amine ...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22884(2-[3-(1H-imidazol-5-yl)propyl]-1-(2-{[(5-methyl-1H...)
Affinity DataKi:  12.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22884(2-[3-(1H-imidazol-5-yl)propyl]-1-(2-{[(5-methyl-1H...)
Affinity DataKi:  19.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM7966([3H]histamine | 2-(1H-imidazol-4-yl)ethan-1-amine ...)
Affinity DataKi:  25.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22904(CHEMBL268229 | Alpha-Methylhistane-R | (2R)-1-(1H-...)
Affinity DataKi:  25.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22888(1-[4-(1H-imidazol-5-yl)butyl]-3-methylthiourea | C...)
Affinity DataKi:  63.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22530(N(alpha)-Methylhistamine | [2-(1H-imidazol-5-yl)et...)
Affinity DataKi:  79.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM7966([3H]histamine | 2-(1H-imidazol-4-yl)ethan-1-amine ...)
Affinity DataKi:  158nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22893(CHEMBL512 | dimethyl[(5-{[(2-{[(E)-1-(methylamino)...)
Affinity DataKi:  5.01E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22567(CHEMBL511 | PYRILAMINE | 3H]pyrilamine | N-[2-(dim...)
Affinity DataKi:  7.94E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22567(CHEMBL511 | PYRILAMINE | 3H]pyrilamine | N-[2-(dim...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Glaxo Research & Development

Curated by PDSP Ki Database
LigandPNGBDBM22893(CHEMBL512 | dimethyl[(5-{[(2-{[(E)-1-(methylamino)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed