Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50006823
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054342(8-{4-[((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  0.246nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054342(8-{4-[((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  0.251nMAssay Description:Displacement of [3H]raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.660nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(3) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  2.74nMAssay Description:Displacement of [3H]raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054338(Butyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  4.42nMAssay Description:Displacement of [3H]raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054333(8-[4-((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2...)
Affinity DataKi:  4.94nMAssay Description:Displacement of [3H]raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054342(8-{4-[((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  4.94nMAssay Description:Displacement of [3H]quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054333(8-[4-((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2...)
Affinity DataKi:  6.46nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50053670(CHEMBL541858 | CHEMBL69985 | ((R)-5-Fluoro-1,2,3,4...)
Affinity DataKi:  8.62nMAssay Description:Displacement of [3H]raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataKi:  13.2nMAssay Description:Displacement of [3H]raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054342(8-{4-[((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  17nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054337(Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  23.8nMAssay Description:Displacement of [3H]raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50053670(CHEMBL541858 | CHEMBL69985 | ((R)-5-Fluoro-1,2,3,4...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054337(Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  28.8nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50053670(CHEMBL541858 | CHEMBL69985 | ((R)-5-Fluoro-1,2,3,4...)
Affinity DataKi:  30.2nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054336(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  35.8nMAssay Description:Displacement of [3H]raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054333(8-[4-((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054338(Butyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  44.5nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054338(Butyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054333(8-[4-((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2...)
Affinity DataKi:  68nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054336(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  108nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054334((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-ylami...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054341(Butyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054336(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  167nMAssay Description:Displacement of [3H]quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054337(Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  179nMAssay Description:Displacement of [3H]quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054335(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  199nMAssay Description:Displacement of [3H]raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50053670(CHEMBL541858 | CHEMBL69985 | ((R)-5-Fluoro-1,2,3,4...)
Affinity DataKi:  201nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054338(Butyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  210nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054341(Butyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  254nMAssay Description:Displacement of [3H]quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054337(Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  415nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054341(Butyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  440nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054339(Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  494nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054334((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-ylami...)
Affinity DataKi:  525nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataKi:  572nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054336(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  582nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054334((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-ylami...)
Affinity DataKi:  585nMAssay Description:Displacement of [3H]quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054340(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  627nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054335(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  644nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054339(Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  779nMAssay Description:Displacement of [3H]quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054341(Butyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  790nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054334((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-ylami...)
Affinity DataKi:  864nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054339(Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [3H]raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054340(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  1.45E+3nMAssay Description:Displacement of [3H]raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054335(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  1.53E+3nMAssay Description:Displacement of [3H]quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054340(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  2.45E+3nMAssay Description:Displacement of [3H]quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054339(Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  2.83E+3nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054335(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  4.72E+3nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054340(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  5.94E+3nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed