Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50041247
TargetIntegrin alpha-V/beta-3(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50237601([5-Benzyl-11-(3-guanidino-propyl)-8-isopropyl-3,6,...)
Affinity DataIC50: 10nMAssay Description:Inhibition of alphaV-beta3 interaction with vitronectinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50369582(DMP-728 | CHEMBL114946)
Affinity DataIC50: 20nMAssay Description:Inhibition of human platelet aggregation mediated by alpha llb/beta3 interaction with fibrinogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50054481((S)-2-[2-((S)-2-{(S)-2-[2-((S)-2-Amino-5-guanidino...)
Affinity DataIC50: 70nMAssay Description:Inhibition of alphaV-beta3 interaction with vitronectinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50054479([(2S,5R,11R,14S)-11-Carboxymethyl-5,14-bis-(3-guan...)
Affinity DataIC50: 140nMAssay Description:Inhibition of alphaV-beta3 interaction with vitronectinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50054478([(2S,5R,11S,14S)-11-Carboxymethyl-5,14-bis-(3-guan...)
Affinity DataIC50: 320nMAssay Description:Inhibition of alphaV-beta3 interaction with vitronectinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50369582(DMP-728 | CHEMBL114946)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of alphaV-beta3 interaction with vitronectinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50054481((S)-2-[2-((S)-2-{(S)-2-[2-((S)-2-Amino-5-guanidino...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human platelet aggregation mediated by alpha llb/beta3 interaction with fibrinogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50237601([5-Benzyl-11-(3-guanidino-propyl)-8-isopropyl-3,6,...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human platelet aggregation mediated by alpha llb/beta3 interaction with fibrinogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50054478([(2S,5R,11S,14S)-11-Carboxymethyl-5,14-bis-(3-guan...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human platelet aggregation mediated by alpha llb/beta3 interaction with fibrinogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50054479([(2S,5R,11R,14S)-11-Carboxymethyl-5,14-bis-(3-guan...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human platelet aggregation mediated by alpha llb/beta3 interaction with fibrinogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed