Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50003445
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Perugia

Curated by ChEMBL
LigandPNGBDBM21690(Ciprinol | 1-cyclopropyl-6-fluoro-4-oxo-7-(piperaz...)
Affinity DataIC50: 2.05E+3nMAssay Description:Inhibitory effect against Escherichia coli Gyrase in Supercoiling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50470984(CHEMBL429961)
Affinity DataIC50: 4.34E+3nMAssay Description:Inhibitory effect against Escherichia coli Gyrase in Supercoiling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50470990(CHEMBL136779)
Affinity DataIC50: 6.96E+3nMAssay Description:Inhibitory effect against Escherichia coli Gyrase in Supercoiling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50470988(CHEMBL141308)
Affinity DataIC50: 7.64E+3nMAssay Description:Inhibitory effect against Escherichia coli Gyrase in Supercoiling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50470986(CHEMBL124970)
Affinity DataIC50: 9.24E+3nMAssay Description:Inhibitory effect against Escherichia coli Gyrase in Supercoiling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50470982(CHEMBL344447)
Affinity DataIC50: 9.37E+3nMAssay Description:Inhibitory effect against Escherichia coli Gyrase in Supercoiling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50470980(CHEMBL145932)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibitory effect against Escherichia coli Gyrase in Supercoiling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50470983(CHEMBL416273)
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibitory effect against Escherichia coli Gyrase in Supercoiling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50470981(CHEMBL343603)
Affinity DataIC50: 1.64E+4nMAssay Description:Inhibitory effect against Escherichia coli Gyrase in Supercoiling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50470987(CHEMBL148052)
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibitory effect against Escherichia coli Gyrase in Supercoiling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50470985(CHEMBL148033)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibitory effect against Escherichia coli Gyrase in Supercoiling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50470979(CHEMBL342273)
Affinity DataIC50: 8.49E+4nMAssay Description:Inhibitory effect against Escherichia coli Gyrase in Supercoiling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50470989(CHEMBL357882 | SQ-4003)
Affinity DataIC50: 9.68E+4nMAssay Description:Inhibitory effect against Escherichia coli Gyrase in Supercoiling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed