Compile Data Set for Download or QSAR
Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 50036585
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.150nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056418(4-Amino-5-chloro-2-methoxy-benzoic acid 2-azepan-1...)
Affinity DataKi:  0.920nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056406(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3-methy...)
Affinity DataKi:  0.930nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056403(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3-hydro...)
Affinity DataKi:  1nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM29526(CHEMBL286136 | 2-Piperidinoethyl 4-amino-5-chloro-...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056416(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-acety...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056411(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-carba...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056424(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-hydro...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056397(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3,3-dim...)
Affinity DataKi:  1.70nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056403(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3-hydro...)
Affinity DataKi:  2nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056392(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3,5-dim...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056392(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3,5-dim...)
Affinity DataKi:  2.32nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056405(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-methy...)
Affinity DataEC50:  3nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056403(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3-hydro...)
Affinity DataEC50:  4nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM29526(CHEMBL286136 | 2-Piperidinoethyl 4-amino-5-chloro-...)
Affinity DataEC50:  4nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056405(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-methy...)
Affinity DataKi:  4.10nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056418(4-Amino-5-chloro-2-methoxy-benzoic acid 2-azepan-1...)
Affinity DataEC50:  4.40nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataEC50:  5nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056409(1-[2-(4-Amino-5-chloro-2-methoxy-benzoyloxy)-ethyl...)
Affinity DataEC50:  5.30nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056412(4-Amino-5-chloro-2-methoxy-benzoic acid 2-pyrrolid...)
Affinity DataKi:  5.40nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056402(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3-aza-b...)
Affinity DataKi:  5.5nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056401(SDZ-205557 | SDZ 205557 | 2-diethylaminoethyl [2-m...)
Affinity DataKi:  5.5nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM48320(SMR000058471 | METOCLOPRAMIDE | METOCLOPRAMIDE HYD...)
Affinity DataEC50:  5.70nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056398(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(2-methy...)
Affinity DataEC50:  6nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056409(1-[2-(4-Amino-5-chloro-2-methoxy-benzoyloxy)-ethyl...)
Affinity DataKi:  6nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056395(1-[2-(4-Amino-5-chloro-2-methoxy-benzoyloxy)-ethyl...)
Affinity DataKi:  6.20nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056422(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(2,6-dim...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056420(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-benzo...)
Affinity DataKi:  7.60nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056398(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(2-methy...)
Affinity DataKi:  7.80nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056402(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3-aza-b...)
Affinity DataEC50:  7.80nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056413(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3,6-dih...)
Affinity DataKi:  9.10nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056400(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(8-aza-b...)
Affinity DataKi:  9.30nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataIC50: 13nMAssay Description:5-hydroxytryptamine 4 receptor antagonist activity, concentration which gave 50% reduction of the 5-HT-induced contractions in the guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056392(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3,5-dim...)
Affinity DataIC50: 13nMAssay Description:5-hydroxytryptamine 4 receptor antagonist activity, concentration which gave 50% reduction of the 5-HT-induced contractions in the guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056416(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-acety...)
Affinity DataEC50:  13nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056424(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-hydro...)
Affinity DataEC50:  14nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056406(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3-methy...)
Affinity DataEC50:  15nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056395(1-[2-(4-Amino-5-chloro-2-methoxy-benzoyloxy)-ethyl...)
Affinity DataEC50:  17nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056411(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-carba...)
Affinity DataEC50:  19nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056421(4-Amino-5-chloro-2-methoxy-benzoic acid 8-methyl-8...)
Affinity DataEC50:  27nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056415(CHEMBL83954 | RS 23597 | 4-Amino-5-chloro-2-methox...)
Affinity DataKi:  28nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056413(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3,6-dih...)
Affinity DataEC50:  29nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056399(4-Amino-5-chloro-2-methoxy-benzoic acid (R)-(1-aza...)
Affinity DataIC50: 30nMAssay Description:5-hydroxytryptamine 4 receptor antagonist activity, concentration which gave 50% reduction of the 5-HT-induced contractions in the guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056415(CHEMBL83954 | RS 23597 | 4-Amino-5-chloro-2-methox...)
Affinity DataEC50:  30nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056414(4-Amino-5-chloro-2-methoxy-benzoic acid 2-morpholi...)
Affinity DataKi:  36nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056412(4-Amino-5-chloro-2-methoxy-benzoic acid 2-pyrrolid...)
Affinity DataEC50:  40nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056400(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(8-aza-b...)
Affinity DataEC50:  40nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056423(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(2,6-dim...)
Affinity DataKi:  40nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056404(BIMU 8 | CHEMBL59834 | 3-Isopropyl-2-oxo-2,3-dihyd...)
Affinity DataEC50:  43nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056407(4-Amino-5-chloro-2-methoxy-benzoic acid 2-dimethyl...)
Affinity DataKi:  47nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
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