Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50036518
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50454555(CHEMBL2115441)
Affinity DataEC50:  0.0980nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058158((3S,6S,9S,12S,15S,18S,26S)-18-((S)-2-Acetylamino-h...)
Affinity DataEC50:  6.10nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058160((3R,6S,9R,12S,15R,18R,26R)-18-Acetylamino-12-benzy...)
Affinity DataEC50:  2.90nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058160((3R,6S,9R,12S,15R,18R,26R)-18-Acetylamino-12-benzy...)
Affinity DataEC50:  89nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50454555(CHEMBL2115441)
Affinity DataEC50:  2.5nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM82411(CAS_75921-69-6 | NDP-MSH)
Affinity DataEC50:  4.10nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058158((3S,6S,9S,12S,15S,18S,26S)-18-((S)-2-Acetylamino-h...)
Affinity DataEC50:  2.61nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058160((3R,6S,9R,12S,15R,18R,26R)-18-Acetylamino-12-benzy...)
Affinity DataEC50:  13nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058161((3S,6R,9S,12S,15S,18R,26S)-18-((S)-2-Acetylamino-h...)
Affinity DataEC50:  3.40nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM82411(CAS_75921-69-6 | NDP-MSH)
Affinity DataEC50:  0.190nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataEC50:  0.190nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataEC50:  1.5nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058161((3S,6R,9S,12S,15S,18R,26S)-18-((S)-2-Acetylamino-h...)
Affinity DataEC50:  34nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058158((3S,6S,9S,12S,15S,18S,26S)-18-((S)-2-Acetylamino-h...)
Affinity DataEC50:  269nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataEC50:  0.240nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataEC50:  0.0400nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM82411(CAS_75921-69-6 | NDP-MSH)
Affinity DataEC50:  0.720nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM82411(CAS_75921-69-6 | NDP-MSH)
Affinity DataEC50:  0.580nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058158((3S,6S,9S,12S,15S,18S,26S)-18-((S)-2-Acetylamino-h...)
Affinity DataEC50:  6.08nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058158((3S,6S,9S,12S,15S,18S,26S)-18-((S)-2-Acetylamino-h...)
Affinity DataEC50:  136nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50454555(CHEMBL2115441)
Affinity DataEC50:  6nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50454555(CHEMBL2115441)
Affinity DataEC50:  28nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataIC50: 0.25nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50454555(CHEMBL2115441)
Affinity DataIC50: 0.350nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM82411(CAS_75921-69-6 | NDP-MSH)
Affinity DataIC50: 0.510nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataIC50: 0.720nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM82411(CAS_75921-69-6 | NDP-MSH)
Affinity DataIC50: 0.860nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50454555(CHEMBL2115441)
Affinity DataIC50: 0.890nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM82411(CAS_75921-69-6 | NDP-MSH)
Affinity DataIC50: 1.20nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM82411(CAS_75921-69-6 | NDP-MSH)
Affinity DataIC50: 1.20nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058160((3R,6S,9R,12S,15R,18R,26R)-18-Acetylamino-12-benzy...)
Affinity DataIC50: 1.90nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058160((3R,6S,9R,12S,15R,18R,26R)-18-Acetylamino-12-benzy...)
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataIC50: 6nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataIC50: 8.60nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058158((3S,6S,9S,12S,15S,18S,26S)-18-((S)-2-Acetylamino-h...)
Affinity DataIC50: 22nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058158((3S,6S,9S,12S,15S,18S,26S)-18-((S)-2-Acetylamino-h...)
Affinity DataIC50: 22.4nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50454555(CHEMBL2115441)
Affinity DataIC50: 25nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50454555(CHEMBL2115441)
Affinity DataIC50: 26nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataIC50: 39nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataIC50: 44nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataIC50: 50nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058158((3S,6S,9S,12S,15S,18S,26S)-18-((S)-2-Acetylamino-h...)
Affinity DataIC50: 72nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058161((3S,6R,9S,12S,15S,18R,26S)-18-((S)-2-Acetylamino-h...)
Affinity DataIC50: 91nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058160((3R,6S,9R,12S,15R,18R,26R)-18-Acetylamino-12-benzy...)
Affinity DataIC50: 102nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058158((3S,6S,9S,12S,15S,18S,26S)-18-((S)-2-Acetylamino-h...)
Affinity DataIC50: 141nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058161((3S,6R,9S,12S,15S,18R,26S)-18-((S)-2-Acetylamino-h...)
Affinity DataIC50: 264nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataIC50: 557nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058160((3R,6S,9R,12S,15R,18R,26R)-18-Acetylamino-12-benzy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058161((3S,6R,9S,12S,15S,18R,26S)-18-((S)-2-Acetylamino-h...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Michigan Medical Center

Curated by ChEMBL
LigandPNGBDBM50058161((3S,6R,9S,12S,15S,18R,26S)-18-((S)-2-Acetylamino-h...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
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