Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50007126
TargetCatechol O-methyltransferase(Pig)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50058814(N,N'-1,3-Propanediylbis(3,4-dihydroxybenzamide) | ...)
Affinity DataKi:  300nMAssay Description:In vitro inhibitory activity against Catechol-O-methyltransferase from porcine liver; Competitive mode of inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCatechol O-methyltransferase(Pig)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50058813(3,4,5-Trihydroxy-N-propyl-benzamide | CHEMBL64275)
Affinity DataKi:  500nMAssay Description:In vitro inhibitory activity against Catechol-O-methyltransferase from porcine liver; Competitive mode of inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCatechol O-methyltransferase(Pig)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50058812(N,N'-1,3-Propanediylbis(3,4,5-trihydroxybenzamide)...)
Affinity DataKi:  6.60E+3nMAssay Description:In vitro inhibitory activity against Catechol-O-methyltransferase from porcine liver; Uncompetitive mode of inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCatechol O-methyltransferase(Pig)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50058815(N,N'-1,5-Pentanediylbis(3,4,5-trihydroxybenzamide)...)
Affinity DataKi:  2.67E+4nMAssay Description:In vitro inhibitory activity against Catechol-O-methyltransferase from porcine liver; Uncompetitive mode of inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCatechol O-methyltransferase(Pig)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50058811(N,N'-1,6-Hexanediylbis(3,4,5-trihydroxybenzamide)H...)
Affinity DataKi:  3.50E+4nMAssay Description:In vitro inhibitory activity against Catechol-O-methyltransferase from porcine liver; Uncompetitive mode of inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCatechol O-methyltransferase(Pig)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50058816(N,N'-1,2-Ethanediylbis(3,4,5-trihydroxybenzamide)H...)
Affinity DataKi:  1.36E+5nMAssay Description:In vitro inhibitory activity against Catechol-O-methyltransferase from porcine liver; Uncompetitive mode of inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed