Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50007179
TargetDelta-type opioid receptor(Mouse)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059367((S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 0.360nMAssay Description:Functional biological activity for Opioid receptor delta 1 was determined in vitro, on mouse vas deferens (MVD).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 0.460nMAssay Description:Functional biological activity for Opioid receptor delta 1 was determined in vitro, on mouse vas deferens (MVD).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059370((S)-3-((S)-2-{2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50: 1.44nMAssay Description:Functional biological activity for Opioid receptor delta 1 was determined in vitro, on mouse vas deferens (MVD).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059367((S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 4.5nMAssay Description:Functional biological activity for mu opioid receptor was determined in vitro, on guinea pig ileum (GPI).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059371((S)-3-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50: 10nMAssay Description:Functional biological activity for mu opioid receptor was determined in vitro, on guinea pig ileum (GPI).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059370((S)-3-((S)-2-{2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50: 10nMAssay Description:Functional biological activity for mu opioid receptor was determined in vitro, on guinea pig ileum (GPI).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059369((R)-3-(2-{2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-prop...)
Affinity DataIC50: 10nMAssay Description:Functional biological activity for mu opioid receptor was determined in vitro, on guinea pig ileum (GPI).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059371((S)-3-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50: 57.3nMAssay Description:Functional biological activity for Opioid receptor delta 1 was determined in vitro, on mouse vas deferens (MVD).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059369((R)-3-(2-{2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-prop...)
Affinity DataIC50: 70nMAssay Description:Functional biological activity for Opioid receptor delta 1 was determined in vitro, on mouse vas deferens (MVD).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 420nMAssay Description:Functional biological activity for mu opioid receptor was determined in vitro, on guinea pig ileum (GPI).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059366(((S)-2-{(S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-h...)
Affinity DataKi:  0.110nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]DPDPE (6.3 nM) for Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059370((S)-3-((S)-2-{2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  0.120nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]DPDPE (6.3 nM) for Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataKi:  0.150nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]DPDPE (6.3 nM) for Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059367((S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-p...)
Affinity DataKi:  0.200nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]DPDPE (6.3 nM) for Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059367((S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-p...)
Affinity DataKi:  0.430nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]- DAGO (1.28 nM) for Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059371((S)-3-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  0.800nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]DPDPE (6.3 nM) for Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059369((R)-3-(2-{2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-prop...)
Affinity DataKi:  3.62nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]DPDPE (6.3 nM) for Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059366(((S)-2-{(S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-h...)
Affinity DataKi:  4.48nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]- DAGO (1.28 nM) for Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059372((S)-3-((R)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  5.72nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]DPDPE (6.3 nM) for Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059373((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  15.5nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]DPDPE (6.3 nM) for Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataKi:  147nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]- DAGO (1.28 nM) for Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059370((S)-3-((S)-2-{2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  1.02E+3nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]- DAGO (1.28 nM) for Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50454611(CHEMBL2370048)
Affinity DataKi:  2.63E+3nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]DPDPE (6.3 nM) for Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059371((S)-3-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  4.54E+3nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]- DAGO (1.28 nM) for Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059373((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  5.40E+3nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]- DAGO (1.28 nM) for Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059372((S)-3-((R)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  1.36E+4nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]- DAGO (1.28 nM) for Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059369((R)-3-(2-{2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-prop...)
Affinity DataKi:  1.52E+4nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]- DAGO (1.28 nM) for Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50454611(CHEMBL2370048)
Affinity DataKi:  4.41E+5nMAssay Description:Affinity was assessed using competitive binding assay labeled with [3H]- DAGO (1.28 nM) for Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed