Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 50007193
Affinity DataIC50: 0.260nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in absence of 120 mM NaCl +...More data for this Ligand-Target Pair
Affinity DataIC50: 0.410nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in absence of 120 mM NaCl +...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in absence of 120 mM NaCl +...More data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in absence of 120 mM NaCl +...More data for this Ligand-Target Pair
Affinity DataIC50: 7.30nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in absence of 120 mM NaCl +...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Affinity against Opioid receptor kappa 2 was determined by measuring the inhibition of [3H]bremazocine binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in presence of 120 mM NaCl ...More data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in absence of 120 mM NaCl +...More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in presence of 120 mM NaCl ...More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in presence of 120 mM NaCl ...More data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in absence of 120 mM NaCl +...More data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in presence of 120 mM NaCl ...More data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in presence of 120 mM NaCl ...More data for this Ligand-Target Pair
Affinity DataIC50: 229nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in presence of 120 mM NaCl ...More data for this Ligand-Target Pair
Affinity DataIC50: 388nMAssay Description:Affinity against Opioid receptor kappa 2 was determined by measuring the inhibition of [3H]bremazocine binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 391nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in presence of 120 mM NaCl ...More data for this Ligand-Target Pair
Affinity DataIC50: 427nMAssay Description:Affinity against Opioid receptor kappa 2 was determined by measuring the inhibition of [3H]bremazocine binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.97E+3nMAssay Description:Affinity against Opioid receptor kappa 2 was determined by measuring the inhibition of [3H]bremazocine binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Affinity against Opioid receptor kappa 1 was determined by measuring the inhibition of [3H]bremazocine binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0290nMAssay Description:Affinity against Opioid receptor kappa 1 was determined by measuring the inhibition of [3H]bremazocine binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Affinity against Opioid receptor kappa 1 was determined by measuring the inhibition of [3H]bremazocine binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0490nMAssay Description:Affinity against Opioid receptor kappa 1 was determined by measuring the inhibition of [3H]bremazocine binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Affinity against Opioid receptor kappa 1 was determined by measuring the inhibition of [3H]bremazocine binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Affinity against Opioid receptor mu 1 was determined by measuring the inhibition of [3H]DAMGO binding to rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Affinity against Opioid receptor kappa 1 was determined by measuring the inhibition of [3H]U-69593 binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Affinity against Opioid receptor delta 1 was determined by measuring the inhibition of [3H]DPDPE binding to rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Affinity against Opioid receptor kappa 1 was determined by measuring the inhibition of [3H]U-69593 binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Affinity against Opioid receptor kappa 1 was determined by measuring the inhibition of [3H]U-69593 binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Affinity against Opioid receptor kappa 1 was determined by measuring the inhibition of [3H]bremazocine binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.66nMAssay Description:Affinity against Opioid receptor kappa 1 was determined by measuring the inhibition of [3H]bremazocine binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Affinity against Opioid receptor mu 1 was determined by measuring the inhibition of [3H]DAMGO binding to rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Affinity against Opioid receptor mu 1 was determined by measuring the inhibition of [3H]DAMGO binding to rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 10.9nMAssay Description:Affinity against Opioid receptor mu 1 was determined by measuring the inhibition of [3H]DAMGO binding to rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Affinity against Opioid receptor kappa 1 was determined by measuring the inhibition of [3H]U-69593 binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Affinity against Opioid receptor kappa 3 was determined by measuring the inhibition of [3H]NalBzoH binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 31.1nMAssay Description:Affinity against Opioid receptor mu 1 was determined by measuring the inhibition of [3H]DAMGO binding to rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 31.7nMAssay Description:Affinity against Opioid receptor mu 1 was determined by measuring the inhibition of [3H]DAMGO binding to rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Affinity against Opioid receptor kappa 3 was determined by measuring the inhibition of [3H]NalBzoH binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Affinity against Opioid receptor kappa 3 was determined by measuring the inhibition of [3H]NalBzoH binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 113nMAssay Description:Affinity against Opioid receptor kappa 3 was determined by measuring the inhibition of [3H]NalBzoH binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 128nMAssay Description:Affinity against Opioid receptor mu 1 was determined by measuring the inhibition of [3H]DAMGO binding to rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 149nMAssay Description:Affinity against Opioid receptor delta 1 was determined by measuring the inhibition of [3H]DPDPE binding to rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 166nMAssay Description:Affinity against Opioid receptor delta 1 was determined by measuring the inhibition of [3H]DPDPE binding to rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 176nMAssay Description:Affinity against Opioid receptor delta 1 was determined by measuring the inhibition of [3H]DPDPE binding to rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 499nMAssay Description:Affinity against Opioid receptor delta 1 was determined by measuring the inhibition of [3H]DPDPE binding to rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 558nMAssay Description:Affinity against Opioid receptor delta 1 was determined by measuring the inhibition of [3H]DPDPE binding to rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.77E+3nMAssay Description:Affinity against Opioid receptor delta 1 was determined by measuring the inhibition of [3H]DPDPE binding to rat forebrain membranesMore data for this Ligand-Target Pair






