Compile Data Set for Download or QSAR
Report error Found 74 Enz. Inhib. hit(s) with all data for entry = 50007261
TargetCholinesterase(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060483(7,8,9,10-Tetrahydro-6H-cyclohepta[b]quinolin-11-yl...)
Affinity DataIC50: 14nMAssay Description:In vitro inhibition of Butyrylcholinesterase from human plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060475(6,7-Dihydro-5H-8-aza-benzo[3,4]cyclohepta[1,2-b]na...)
Affinity DataIC50: 20nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 25nMAssay Description:In vitro inhibition of Butyrylcholinesterase from human plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholinesterase(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060483(7,8,9,10-Tetrahydro-6H-cyclohepta[b]quinolin-11-yl...)
Affinity DataIC50: 39nMAssay Description:In vitro inhibition of acetylcholinesterase, isolated from rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060470(10-azoniatetracyclo[10.2.1.02,11.04,9]pentadeca-2,...)
Affinity DataIC50: 41nMAssay Description:In vitro inhibition of Butyrylcholinesterase from human plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060477(2,3-dihydro-1H-cyclopenta[b]quinolin-9-amine | 2,3...)
Affinity DataIC50: 52nMAssay Description:In vitro inhibition of Butyrylcholinesterase from human plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060477(2,3-dihydro-1H-cyclopenta[b]quinolin-9-amine | 2,3...)
Affinity DataIC50: 56nMAssay Description:In vitro inhibition of acetylcholinesterase, isolated from rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 78nMAssay Description:In vitro inhibition of acetylcholinesterase, isolated from rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM30130(Prozac | cid_62857 | Fluoxetin | CHEMBL41 | CHEMBL...)
Affinity DataIC50: 130nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060470(10-azoniatetracyclo[10.2.1.02,11.04,9]pentadeca-2,...)
Affinity DataIC50: 200nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060479(3-chlorodibenzo[b,h][1,6]naphthyridin-7-amine | 3-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of neuronal uptake of Noradrenaline in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060470(10-azoniatetracyclo[10.2.1.02,11.04,9]pentadeca-2,...)
Affinity DataIC50: 240nMAssay Description:In vitro inhibition of acetylcholinesterase, isolated from rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM9074(CHEMBL60167 | 10H-indeno[1,2-b]quinolin-11-amine |...)
Affinity DataIC50: 350nMAssay Description:In vitro inhibition of acetylcholinesterase, isolated from rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060477(2,3-dihydro-1H-cyclopenta[b]quinolin-9-amine | 2,3...)
Affinity DataIC50: 600nMAssay Description:Inhibition of neuronal uptake of Noradrenaline in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060474(3-Methoxy-6,7-dihydro-5H-13-aza-benzo[3,4]cyclohep...)
Affinity DataIC50: 700nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060472(6,7,8,9,10,11-hexahydrocycloocta[b]quinolin-12-ami...)
Affinity DataIC50: 800nMAssay Description:Inhibition of neuronal uptake of Noradrenaline in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060472(6,7,8,9,10,11-hexahydrocycloocta[b]quinolin-12-ami...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060478(3-Methoxy-5,6-dihydro-benzo[c]acridin-7-ylamine | ...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of neuronal uptake of Noradrenaline in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM35229(Desmethylimipramine | 3-(10,11-dihydro-5H-dibenzo[...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of neuronal uptake of Noradrenaline in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTransporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060473(6,7-Dihydro-5H-13-aza-benzo[3,4]cyclohepta[1,2-b]n...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of neuronal uptake of Noradrenaline in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM9074(CHEMBL60167 | 10H-indeno[1,2-b]quinolin-11-amine |...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM9074(CHEMBL60167 | 10H-indeno[1,2-b]quinolin-11-amine |...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of neuronal uptake of Noradrenaline in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060472(6,7,8,9,10,11-hexahydrocycloocta[b]quinolin-12-ami...)
Affinity DataIC50: 2.30E+3nMAssay Description:In vitro inhibition of Butyrylcholinesterase from human plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060476(5,6,7,8-tetrahydrobenzo[2,3]azocino[4,5-b]quinolin...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of neuronal uptake of Noradrenaline in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060485(6,7-Dihydro-5H-benzo[2,3]azepino[4,5-b]quinolin-8-...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of neuronal uptake of Noradrenaline in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM9074(CHEMBL60167 | 10H-indeno[1,2-b]quinolin-11-amine |...)
Affinity DataIC50: 3.10E+3nMAssay Description:In vitro inhibition of Butyrylcholinesterase from human plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060481(5,6-dihydrobenzo[c]acridin-7-amine | 5,6-Dihydro-b...)
Affinity DataIC50: 3.30E+3nMAssay Description:In vitro inhibition of Butyrylcholinesterase from human plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060469(2,3-dimethyl-1H-cyclopenta[b]quinolin-9-amine | 2,...)
Affinity DataIC50: 3.50E+3nMAssay Description:In vitro inhibition of acetylcholinesterase, isolated from rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060483(7,8,9,10-Tetrahydro-6H-cyclohepta[b]quinolin-11-yl...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060474(3-Methoxy-6,7-dihydro-5H-13-aza-benzo[3,4]cyclohep...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of neuronal uptake of Noradrenaline in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060485(6,7-Dihydro-5H-benzo[2,3]azepino[4,5-b]quinolin-8-...)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060480(9-Amino-2,3-dimethyl-2,3-dihydro-1H-cyclopenta[b]q...)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060481(5,6-dihydrobenzo[c]acridin-7-amine | 5,6-Dihydro-b...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060473(6,7-Dihydro-5H-13-aza-benzo[3,4]cyclohepta[1,2-b]n...)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060469(2,3-dimethyl-1H-cyclopenta[b]quinolin-9-amine | 2,...)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060478(3-Methoxy-5,6-dihydro-benzo[c]acridin-7-ylamine | ...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060469(2,3-dimethyl-1H-cyclopenta[b]quinolin-9-amine | 2,...)
Affinity DataIC50: 5.90E+3nMAssay Description:In vitro inhibition of Butyrylcholinesterase from human plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060470(10-azoniatetracyclo[10.2.1.02,11.04,9]pentadeca-2,...)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of neuronal uptake of Noradrenaline in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060476(5,6,7,8-tetrahydrobenzo[2,3]azocino[4,5-b]quinolin...)
Affinity DataIC50: 6.70E+3nMAssay Description:In vitro inhibition of Butyrylcholinesterase from human plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060476(5,6,7,8-tetrahydrobenzo[2,3]azocino[4,5-b]quinolin...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060483(7,8,9,10-Tetrahydro-6H-cyclohepta[b]quinolin-11-yl...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of neuronal uptake of Noradrenaline in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060484(9-Amino-3-butyl-2-methyl-2,3-dihydro-1H-cyclopenta...)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of neuronal uptake of Noradrenaline in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060472(6,7,8,9,10,11-hexahydrocycloocta[b]quinolin-12-ami...)
Affinity DataIC50: 9.10E+3nMAssay Description:In vitro inhibition of acetylcholinesterase, isolated from rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060471(4-Chloro-5,6-dihydro-benzo[c]acridin-7-ylamine | C...)
Affinity DataIC50: 1.03E+4nMAssay Description:In vitro inhibition of Butyrylcholinesterase from human plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060484(9-Amino-3-butyl-2-methyl-2,3-dihydro-1H-cyclopenta...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of neuronal uptake of Noradrenaline in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060481(5,6-dihydrobenzo[c]acridin-7-amine | 5,6-Dihydro-b...)
Affinity DataIC50: 1.21E+4nMAssay Description:Inhibition of neuronal uptake of Noradrenaline in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060480(9-Amino-2,3-dimethyl-2,3-dihydro-1H-cyclopenta[b]q...)
Affinity DataIC50: 1.22E+4nMAssay Description:In vitro inhibition of Butyrylcholinesterase from human plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50060486(3-butyl-2-methyl-1H-cyclopenta[b]quinolin-9-amine ...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of neuronal uptake of 5 - Hydroxytryptamine in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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