Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50007540
TargetGABA A receptor alpha-1/beta-1/gamma-2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50064417(4-Bromo-2,6-diisopropyl-phenol | CHEMBL54497)
Affinity DataEC50:  3.80E+4nMAssay Description:Direct activation of chloride current in Xenopus laevis oocytes expressing human alpha-1-beta-1-gamma-2 GABA-A receptor subunitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGABA A receptor alpha-1/beta-1/gamma-2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50058046(propofol | CHEMBL526)
Affinity DataEC50:  4.40E+4nMAssay Description:Direct activation of chloride current in Xenopus laevis oocytes expressing human alpha-1-beta-1-gamma-2 GABA-A receptor subunitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGABA A receptor alpha-1/beta-1/gamma-2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50064420((4-Hydroxy-3,5-diisopropyl-phenyl)-phenyl-methanon...)
Affinity DataEC50:  4.70E+4nMAssay Description:Direct activation of chloride current in Xenopus laevis oocytes expressing human alpha-1-beta-1-gamma-2 GABA-A receptor subunitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGABA A receptor alpha-1/beta-1/gamma-2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50064419(4-Chloro-2,6-diisopropyl-phenol | CHEMBL292402)
Affinity DataEC50:  1.00E+4nMAssay Description:Modulation of GABA-induced chloride currents in Xenopus laevis oocytes expressing human alpha-1-beta-1-gamma-2 GABA-A receptor subunitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGABA A receptor alpha-1/beta-1/gamma-2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50064424(4-Iodo-2,6-diisopropylphenol | 4-Iodo-2,6-diisopro...)
Affinity DataEC50:  1.20E+4nMAssay Description:Modulation of GABA-induced chloride currents in Xenopus laevis oocytes expressing human alpha-1-beta-1-gamma-2 GABA-A receptor subunitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGABA A receptor alpha-1/beta-1/gamma-2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50058046(propofol | CHEMBL526)
Affinity DataEC50:  8.00E+3nMAssay Description:Modulation of GABA-induced chloride currents in Xenopus laevis oocytes expressing human alpha-1-beta-1-gamma-2 GABA-A receptor subunitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGABA A receptor alpha-1/beta-1/gamma-2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50064417(4-Bromo-2,6-diisopropyl-phenol | CHEMBL54497)
Affinity DataEC50:  1.20E+4nMAssay Description:Modulation of GABA-induced chloride currents in Xenopus laevis oocytes expressing human alpha-1-beta-1-gamma-2 GABA-A receptor subunitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGABA A receptor alpha-1/beta-1/gamma-2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50064424(4-Iodo-2,6-diisopropylphenol | 4-Iodo-2,6-diisopro...)
Affinity DataEC50:  5.10E+4nMAssay Description:Direct activation of chloride current in Xenopus laevis oocytes expressing human alpha-1-beta-1-gamma-2 GABA-A receptor subunitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGABA A receptor alpha-1/beta-1/gamma-2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50064420((4-Hydroxy-3,5-diisopropyl-phenyl)-phenyl-methanon...)
Affinity DataEC50:  9.00E+3nMAssay Description:Modulation of GABA-induced chloride currents in Xenopus laevis oocytes expressing human alpha-1-beta-1-gamma-2 GABA-A receptor subunitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGABA A receptor alpha-1/beta-1/gamma-2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50064419(4-Chloro-2,6-diisopropyl-phenol | CHEMBL292402)
Affinity DataEC50:  3.80E+4nMAssay Description:Direct activation of chloride current in Xenopus laevis oocytes expressing human alpha-1-beta-1-gamma-2 GABA-A receptor subunitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed