Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50036619
TargetDipeptidyl peptidase 4(Human)
University of Versailles Saint-Quentin-en-Yvelines

Curated by ChEMBL
LigandPNGBDBM50064660(Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SMe2]-Gly4-), 2CF3...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by CD26 (Dipeptidyl peptidase IV) purified from CEM H01 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Versailles Saint-Quentin-en-Yvelines

Curated by ChEMBL
LigandPNGBDBM50064657(Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SMe2+]-Gly2-), 2CF...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by CD26 (Dipeptidyl peptidase IV) purified from CEM H01 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Versailles Saint-Quentin-en-Yvelines

Curated by ChEMBL
LigandPNGBDBM50064661(Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SBu2]-Gly2-), 2CF3...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by CD26 (Dipeptidyl peptidase IV) purified from CEM H01 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Versailles Saint-Quentin-en-Yvelines

Curated by ChEMBL
LigandPNGBDBM50064656(Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SOct2-]-Gly2-), 2C...)
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by CD26 (Dipeptidyl peptidase IV) purified from CEM H01 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Versailles Saint-Quentin-en-Yvelines

Curated by ChEMBL
LigandPNGBDBM50064661(Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SBu2]-Gly2-), 2CF3...)
Affinity DataIC50: 570nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by Dipeptidyl peptidase IV purified from CD26-negative C8166 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Versailles Saint-Quentin-en-Yvelines

Curated by ChEMBL
LigandPNGBDBM50064660(Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SMe2]-Gly4-), 2CF3...)
Affinity DataIC50: 610nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by Dipeptidyl peptidase IV purified from CD26-negative C8166 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Versailles Saint-Quentin-en-Yvelines

Curated by ChEMBL
LigandPNGBDBM50064656(Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SOct2-]-Gly2-), 2C...)
Affinity DataIC50: 630nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by Dipeptidyl peptidase IV purified from CD26-negative C8166 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Versailles Saint-Quentin-en-Yvelines

Curated by ChEMBL
LigandPNGBDBM50064657(Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SMe2+]-Gly2-), 2CF...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by Dipeptidyl peptidase IV purified from CD26-negative C8166 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Versailles Saint-Quentin-en-Yvelines

Curated by ChEMBL
LigandPNGBDBM50064658(Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2OAc]-Gly2-), CF3CO...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by CD26 (Dipeptidyl peptidase IV) purified from CEM H01 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Versailles Saint-Quentin-en-Yvelines

Curated by ChEMBL
LigandPNGBDBM50064658(Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2OAc]-Gly2-), CF3CO...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by Dipeptidyl peptidase IV purified from CD26-negative C8166 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Versailles Saint-Quentin-en-Yvelines

Curated by ChEMBL
LigandPNGBDBM50064659((4S,10S)-10-Amino-24-phenoxymethyl-2,8,15,18,21-pe...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by CD26 (Dipeptidyl peptidase IV) purified from CEM H01 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Versailles Saint-Quentin-en-Yvelines

Curated by ChEMBL
LigandPNGBDBM50064659((4S,10S)-10-Amino-24-phenoxymethyl-2,8,15,18,21-pe...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by Dipeptidyl peptidase IV purified from CD26-negative C8166 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Versailles Saint-Quentin-en-Yvelines

Curated by ChEMBL
LigandPNGBDBM50064657(Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SMe2+]-Gly2-), 2CF...)
Affinity DataKi:  85nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by CD26 (dipeptidylpeptidase 4) purified from CEM H01 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Versailles Saint-Quentin-en-Yvelines

Curated by ChEMBL
LigandPNGBDBM50064657(Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SMe2+]-Gly2-), 2CF...)
Affinity DataKi:  470nMAssay Description:Inhibitory kinetic constant against Dipeptidyl peptidase IV purified from CD26-negative C8166 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed