Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50036624
TargetPepsin A-5(Human)
Institute of Pharmaceutical Chemistry

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 59nMAssay Description:Inhibitory activity against pepsin as oxidation of o-phenylenediamine by Horse radish peroxidase (Pepsin sensitive)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetPepsin A-5(Human)
Institute of Pharmaceutical Chemistry

Curated by ChEMBL
LigandPNGBDBM50064908({1-[1-((S)-2-Hydroxy-1-propyl-octylcarbamoyl)-2-me...)
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against pepsin as oxidation of o-phenylenediamine by Horse radish peroxidase (Pepsin sensitive)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetPepsin A-5(Human)
Institute of Pharmaceutical Chemistry

Curated by ChEMBL
LigandPNGBDBM50064905({1-[1-((S)-2-Hydroxy-1-isobutyl-decylcarbamoyl)-2-...)
Affinity DataIC50: 790nMAssay Description:Inhibitory activity against pepsin as oxidation of o-phenylenediamine by Horse radish peroxidase (Pepsin sensitive)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetPepsin A-5(Human)
Institute of Pharmaceutical Chemistry

Curated by ChEMBL
LigandPNGBDBM50064912({1-[1-((S)-2-Hydroxy-1-isobutyl-octylcarbamoyl)-2-...)
Affinity DataIC50: 830nMAssay Description:Inhibitory activity against pepsin as oxidation of o-phenylenediamine by Horse radish peroxidase (Pepsin sensitive)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetPepsin A-5(Human)
Institute of Pharmaceutical Chemistry

Curated by ChEMBL
LigandPNGBDBM50064909({1-[1-((S)-2-Hydroxy-1-propyl-hexylcarbamoyl)-2-me...)
Affinity DataIC50: 910nMAssay Description:Inhibitory activity against pepsin as oxidation of o-phenylenediamine by Horse radish peroxidase (Pepsin sensitive)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetPepsin A-5(Human)
Institute of Pharmaceutical Chemistry

Curated by ChEMBL
LigandPNGBDBM50064911({1-[1-((S)-2-Hydroxy-1-propyl-decylcarbamoyl)-2-me...)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibitory activity against pepsin as oxidation of o-phenylenediamine by Horse radish peroxidase (Pepsin sensitive)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetPepsin A-5(Human)
Institute of Pharmaceutical Chemistry

Curated by ChEMBL
LigandPNGBDBM50064910({1-[1-((S)-2-Hydroxy-1-isobutyl-hexylcarbamoyl)-2-...)
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibitory activity against pepsin as oxidation of o-phenylenediamine by Horse radish peroxidase (Pepsin sensitive)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetPepsin A-5(Human)
Institute of Pharmaceutical Chemistry

Curated by ChEMBL
LigandPNGBDBM50064906({1-[1-((S)-1-sec-Butyl-2-hydroxy-decylcarbamoyl)-2...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against pepsin as oxidation of o-phenylenediamine by Horse radish peroxidase (Pepsin sensitive)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetPepsin A-5(Human)
Institute of Pharmaceutical Chemistry

Curated by ChEMBL
LigandPNGBDBM50064907({1-[1-((S)-1-sec-Butyl-2-hydroxy-octylcarbamoyl)-2...)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibitory activity against pepsin as oxidation of o-phenylenediamine by Horse radish peroxidase (Pepsin sensitive)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetPepsin A-5(Human)
Institute of Pharmaceutical Chemistry

Curated by ChEMBL
LigandPNGBDBM50369360(CHEMBL1790562)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibitory activity against pepsin as oxidation of o-phenylenediamine by Horse radish peroxidase (Pepsin sensitive)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed