Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50007611
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065348((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(2-oxo-...)
Affinity DataIC50: 250nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065336((1S,4aS,5R)-1,4a-Dimethyl-6-oxo-5-[2-(2-oxo-2,5-di...)
Affinity DataIC50: 260nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065344(methyl 5,8a-dimethyl-1-[2-(2-oxo-2,5-dihydro-3-fur...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065343((1S,4aR,5S,6S)-6-Hydroxymethyl-1,4a-dimethyl-5-[2-...)
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065347(3-[2-((1S,5S,8aR)-5-Methoxymethyl-5,8a-dimethyl-2-...)
Affinity DataIC50: 1.70E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065339((1S,4aS)-6-Formyl-1,4a-dimethyl-5-[2-(2-oxo-2,5-di...)
Affinity DataIC50: 1.70E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065352((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(2-oxo-...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065335((1S,4aS,5R,6S)-6-Hydroxy-1,4a-dimethyl-5-[2-(2-oxo...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065342((1S,4aS,5R)-1,4a-Dimethyl-6-oxo-5-[2-(2-oxo-tetrah...)
Affinity DataIC50: 2.60E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065333(6-Hydroxymethyl-1,4a-dimethyl-5-[2-(2-oxo-2,5-dihy...)
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065345((1S,4aR,5S)-1,4a,6-Trimethyl-5-[2-(2-oxo-tetrahydr...)
Affinity DataIC50: 4.80E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065346((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(5-oxo-...)
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065341((1R,6S,9aS)-6,9a-Dimethyl-3-oxo-1-[2-(5-oxo-2,5-di...)
Affinity DataIC50: 8.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065337((1S,4aR,5S)-5-((Z)-5-Hydroxy-3-hydroxymethyl-pent-...)
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065351((Z)-2-[2-((1S,5S,8aR)-5-Hydroxymethyl-5,8a-dimethy...)
Affinity DataIC50: 2.10E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065350((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(2-oxo-...)
Affinity DataIC50: 2.30E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065338(3-[2-((1S,5S,8aR)-5-Hydroxymethyl-5,8a-dimethyl-2-...)
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065349(4-[2-((1S,5S,8aR)-5-Hydroxymethyl-5,8a-dimethyl-2-...)
Affinity DataIC50: 1.10E+5nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065340((1S,4aR,5S)-5-(2-Furan-3-yl-ethyl)-1,4a-dimethyl-6...)
Affinity DataIC50: 1.00E+6nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065334((1S,4aS,5R,6R)-6-Hydroxy-6-hydroxymethyl-1,4a-dime...)
Affinity DataIC50: 1.00E+6nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed