Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50036650
TargetMu-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066532(1N-[4-cyclopropylmethyl-14-oxo-10-(2-propynyloxy)-...)
Affinity DataKi:  1.60nMAssay Description:In vitro binding affinity against Opioid receptor mu 1 (DAMGO) opioid receptor in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50195656(clocinnamox | 1N-[4-cyclopropylmethyl-10-hydroxy-1...)
Affinity DataKi:  5.40nMAssay Description:In vitro binding affinity against Opioid receptor kappa 1 in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066531(methyl 2-[17-[2-(4-chlorophenyl)-(E)-1-ethenylcarb...)
Affinity DataKi:  7.60nMAssay Description:In vitro binding affinity against Opioid receptor mu 1 (DAMGO) opioid receptor in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066536(1N-[10-cyclopropylmethoxy-4-cyclopropylmethyl-14-o...)
Affinity DataKi:  7.60nMAssay Description:In vitro binding affinity against Opioid receptor mu 1 (DAMGO) opioid receptor in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066534(1N-[10-allyloxy-4-cyclopropylmethyl-14-oxo-(17S)-1...)
Affinity DataKi:  8.90nMAssay Description:In vitro binding affinity against Opioid receptor mu 1 (DAMGO) opioid receptor in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50195656(clocinnamox | 1N-[4-cyclopropylmethyl-10-hydroxy-1...)
Affinity DataKi:  9nMAssay Description:In vitro binding affinity against Opioid receptor mu 1 (DAMGO) opioid receptor in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066533(1N-[10-cyanomethoxy-4-cyclopropylmethyl-14-oxo-(17...)
Affinity DataKi:  12nMAssay Description:In vitro binding affinity against Opioid receptor mu 1 (DAMGO) opioid receptor in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50195656(clocinnamox | 1N-[4-cyclopropylmethyl-10-hydroxy-1...)
Affinity DataKi:  13nMAssay Description:In vitro binding affinity against Opioid receptor delta 1 (DPDPE) in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066530(1N-[4-cyclopropylmethyl-10-isopropoxy-14-oxo-(17S)...)
Affinity DataKi:  15nMAssay Description:In vitro binding affinity against Opioid receptor kappa 1 in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066533(1N-[10-cyanomethoxy-4-cyclopropylmethyl-14-oxo-(17...)
Affinity DataKi:  18nMAssay Description:In vitro binding affinity against Opioid receptor kappa 1 in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066534(1N-[10-allyloxy-4-cyclopropylmethyl-14-oxo-(17S)-1...)
Affinity DataKi:  18nMAssay Description:In vitro binding affinity against Opioid receptor kappa 1 in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066537(1N-[4-cyclopropylmethyl-14-oxo-10-propoxy-(17S)-12...)
Affinity DataKi:  19nMAssay Description:In vitro binding affinity against Opioid receptor kappa 1 in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066532(1N-[4-cyclopropylmethyl-14-oxo-10-(2-propynyloxy)-...)
Affinity DataKi:  19nMAssay Description:In vitro binding affinity against Opioid receptor kappa 1 in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066532(1N-[4-cyclopropylmethyl-14-oxo-10-(2-propynyloxy)-...)
Affinity DataKi:  21nMAssay Description:In vitro binding affinity against Opioid receptor delta 1 (DPDPE) in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066531(methyl 2-[17-[2-(4-chlorophenyl)-(E)-1-ethenylcarb...)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity against Opioid receptor delta 1 (DPDPE) in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066537(1N-[4-cyclopropylmethyl-14-oxo-10-propoxy-(17S)-12...)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity against Opioid receptor mu 1 (DAMGO) opioid receptor in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066536(1N-[10-cyclopropylmethoxy-4-cyclopropylmethyl-14-o...)
Affinity DataKi:  57nMAssay Description:In vitro binding affinity against Opioid receptor delta 1 (DPDPE) in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066530(1N-[4-cyclopropylmethyl-10-isopropoxy-14-oxo-(17S)...)
Affinity DataKi:  60nMAssay Description:In vitro binding affinity against Opioid receptor mu 1 (DAMGO) opioid receptor in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066534(1N-[10-allyloxy-4-cyclopropylmethyl-14-oxo-(17S)-1...)
Affinity DataKi:  65nMAssay Description:In vitro binding affinity against Opioid receptor delta 1 (DPDPE) in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066537(1N-[4-cyclopropylmethyl-14-oxo-10-propoxy-(17S)-12...)
Affinity DataKi:  83nMAssay Description:In vitro binding affinity against Opioid receptor delta 1 (DPDPE) in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066533(1N-[10-cyanomethoxy-4-cyclopropylmethyl-14-oxo-(17...)
Affinity DataKi:  90nMAssay Description:In vitro binding affinity against Opioid receptor delta 1 (DPDPE) in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066531(methyl 2-[17-[2-(4-chlorophenyl)-(E)-1-ethenylcarb...)
Affinity DataKi:  95nMAssay Description:In vitro binding affinity against Opioid receptor kappa 1 in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066530(1N-[4-cyclopropylmethyl-10-isopropoxy-14-oxo-(17S)...)
Affinity DataKi:  96nMAssay Description:In vitro binding affinity against Opioid receptor delta 1 (DPDPE) in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50066536(1N-[10-cyclopropylmethoxy-4-cyclopropylmethyl-14-o...)
Affinity DataKi:  131nMAssay Description:In vitro binding affinity against Opioid receptor kappa 1 in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed