Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50041265
TargetMuscarinic acetylcholine receptor M2(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM82423(NSC_132947 | CAS_132947 | TRIPITRAMINE)
Affinity DataKi:  0.300nMAssay Description:Inhibition of [3H]NMS binding to rat heart Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408535(CHEMBL131865)
Affinity DataKi:  0.370nMAssay Description:Inhibition of [3H]NMS binding to rat heart Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408530(CHEMBL1202003)
Affinity DataKi:  0.440nMAssay Description:Inhibition of [3H]NMS binding to rat heart Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408535(CHEMBL131865)
Affinity DataKi:  0.5nMAssay Description:Binding affinity for rat cortex Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408527(CHEMBL1202004)
Affinity DataKi:  0.560nMAssay Description:Inhibition of [3H]NMS binding to rat heart Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408525(CHEMBL1202000)
Affinity DataKi:  0.910nMAssay Description:Inhibition of [3H]NMS binding to rat heart Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408530(CHEMBL1202003)
Affinity DataKi:  0.950nMAssay Description:Binding affinity for rat cortex Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408535(CHEMBL131865)
Affinity DataKi:  1.40nMAssay Description:Inhibition of NG 108-15 binding to Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408539(CHEMBL407678)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [3H]NMS binding to rat heart Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408527(CHEMBL1202004)
Affinity DataKi:  2.80nMAssay Description:Inhibition of NG 108-15 binding to Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408535(CHEMBL131865)
Affinity DataKi:  3nMAssay Description:Inhibition of [3H]NMS binding to rat submaxillary gland Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM82423(NSC_132947 | CAS_132947 | TRIPITRAMINE)
Affinity DataKi:  3.5nMAssay Description:Binding affinity for rat cortex Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50407222(CHEMBL112244)
Affinity DataKi:  4.40nMAssay Description:Binding affinity for rat cortex Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408532(CHEMBL134692)
Affinity DataKi:  5.60nMAssay Description:Inhibition of [3H]NMS binding to rat heart Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50407222(CHEMBL112244)
Affinity DataKi:  7.80nMAssay Description:Inhibition of [3H]NMS binding to rat heart Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408533(CHEMBL1202002)
Affinity DataKi:  9.30nMAssay Description:Inhibition of [3H]NMS binding to rat heart Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM82423(NSC_132947 | CAS_132947 | TRIPITRAMINE)
Affinity DataKi:  11nMAssay Description:Inhibition of NG 108-15 binding to Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408525(CHEMBL1202000)
Affinity DataKi:  13nMAssay Description:Binding affinity for rat cortex Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408529(CHEMBL1202001)
Affinity DataKi:  14nMAssay Description:Binding affinity for rat cortex Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408527(CHEMBL1202004)
Affinity DataKi:  15nMAssay Description:Binding affinity for rat cortex Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50407222(CHEMBL112244)
Affinity DataKi:  16nMAssay Description:Inhibition of NG 108-15 binding to Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50064176(METHOCTRAMINE | N,N''-Bis-[6-(2-methoxy-benzylamin...)
Affinity DataKi:  20nMAssay Description:Inhibition of [3H]NMS binding to rat heart Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408540(CHEMBL335115)
Affinity DataKi:  20nMAssay Description:Inhibition of NG 108-15 binding to Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408529(CHEMBL1202001)
Affinity DataKi:  21nMAssay Description:Inhibition of [3H]NMS binding to rat heart Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408533(CHEMBL1202002)
Affinity DataKi:  25nMAssay Description:Binding affinity for rat cortex Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50064176(METHOCTRAMINE | N,N''-Bis-[6-(2-methoxy-benzylamin...)
Affinity DataKi:  32nMAssay Description:Inhibition of NG 108-15 binding to Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408529(CHEMBL1202001)
Affinity DataKi:  36nMAssay Description:Inhibition of NG 108-15 binding to Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408525(CHEMBL1202000)
Affinity DataKi:  40nMAssay Description:Inhibition of NG 108-15 binding to Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408530(CHEMBL1202003)
Affinity DataKi:  42nMAssay Description:Inhibition of NG 108-15 binding to Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50064176(METHOCTRAMINE | N,N''-Bis-[6-(2-methoxy-benzylamin...)
Affinity DataKi:  42nMAssay Description:Binding affinity for rat cortex Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408540(CHEMBL335115)
Affinity DataKi:  45nMAssay Description:Inhibition of [3H]NMS binding to rat heart Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408539(CHEMBL407678)
Affinity DataKi:  50nMAssay Description:Binding affinity for rat cortex Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408532(CHEMBL134692)
Affinity DataKi:  63nMAssay Description:Binding affinity for rat cortex Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408532(CHEMBL134692)
Affinity DataKi:  63nMAssay Description:Inhibition of NG 108-15 binding to Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408532(CHEMBL134692)
Affinity DataKi:  71nMAssay Description:Inhibition of [3H]NMS binding to rat submaxillary gland Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408530(CHEMBL1202003)
Affinity DataKi:  110nMAssay Description:Inhibition of [3H]NMS binding to rat submaxillary gland Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408527(CHEMBL1202004)
Affinity DataKi:  115nMAssay Description:Inhibition of [3H]NMS binding to rat submaxillary gland Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM82423(NSC_132947 | CAS_132947 | TRIPITRAMINE)
Affinity DataKi:  148nMAssay Description:Inhibition of [3H]NMS binding to rat submaxillary gland Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408540(CHEMBL335115)
Affinity DataKi:  158nMAssay Description:Inhibition of [3H]NMS binding to rat submaxillary gland Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408533(CHEMBL1202002)
Affinity DataKi:  158nMAssay Description:Inhibition of NG 108-15 binding to Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408539(CHEMBL407678)
Affinity DataKi:  158nMAssay Description:Inhibition of NG 108-15 binding to Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408540(CHEMBL335115)
Affinity DataKi:  316nMAssay Description:Binding affinity for rat cortex Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50407222(CHEMBL112244)
Affinity DataKi:  331nMAssay Description:Inhibition of [3H]NMS binding to rat submaxillary gland Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408525(CHEMBL1202000)
Affinity DataKi:  398nMAssay Description:Inhibition of [3H]NMS binding to rat submaxillary gland Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50064176(METHOCTRAMINE | N,N''-Bis-[6-(2-methoxy-benzylamin...)
Affinity DataKi:  955nMAssay Description:Inhibition of [3H]NMS binding to rat submaxillary gland Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408533(CHEMBL1202002)
Affinity DataKi:  2.51E+3nMAssay Description:Inhibition of [3H]NMS binding to rat submaxillary gland Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408529(CHEMBL1202001)
Affinity DataKi:  2.57E+3nMAssay Description:Inhibition of [3H]NMS binding to rat submaxillary gland Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50408539(CHEMBL407678)
Affinity DataKi:  5.75E+3nMAssay Description:Inhibition of [3H]NMS binding to rat submaxillary gland Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed