Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50036677
LigandPNGBDBM50067848((S)-2-[(3aR,6R,9S)-3-(1,5-Dimethyl-hexyl)-3a,6,9-t...)
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067843(2-[3-(1,5-Dimethyl-hexyl)-3a,6-dimethyl-7-oxo-dode...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50250718(Clavaric acid | 2-alpha-(3'-hydroxy-3'-methylgluta...)
Affinity DataIC50: 350nMAssay Description:Inhibition of human Farnesyltransferase using Ras-CVLSMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067852(3-[3-(1,5-Dimethyl-hexyl)-3a,6,9-trimethyl-7-oxo-d...)
Affinity DataIC50: 900nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067825(3-[(R)-3-(1,5-Dimethyl-hexyl)-3a-methyl-7-oxo-dode...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067842(2'',15''-dimethyl-5'',17''-dioxo-(2''R,5'R,15''S)-...)
Affinity DataIC50: 1.20E+3nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50250718(Clavaric acid | 2-alpha-(3'-hydroxy-3'-methylgluta...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human Farnesyltransferase using Ras-CVIMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067849((S)-2-[(3aR,6R,9S)-3-(1,5-Dimethyl-hexyl)-9-ethyl-...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067854(Isobutyric acid 2-((10R,13S)-10,13-dimethyl-3,11-d...)
Affinity DataIC50: 6.80E+3nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067834((3aR,6R)-6-(2-Carboxy-ethyl)-3-(1,5-dimethyl-hexyl...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067835((10S,13R,14R)-17-(1,5-Dimethyl-hex-4-enyl)-4,4,10,...)
Affinity DataIC50: 1.20E+4nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50455157(Cortisone | Cortisone acetate | Cortone)
Affinity DataIC50: 1.40E+4nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067846((2R,10S,13R,14R,17R)-17-((R)-4,5-Dihydroxy-1,5-dim...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human Farnesyltransferase using Ras-CVLSMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067841(Isobutyric acid 2-((10R,13S,17R)-17-hydroxy-10,13-...)
Affinity DataIC50: 1.50E+4nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067846((2R,10S,13R,14R,17R)-17-((R)-4,5-Dihydroxy-1,5-dim...)
Affinity DataIC50: 1.50E+4nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067830((3aR,6R,7R)-6-(2-Carboxy-ethyl)-3-(1,5-dimethyl-he...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067831(Succinic acid mono-[2-((10R,13S)-17-hydroxy-10,13-...)
Affinity DataIC50: 2.40E+4nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067851(methyl 3-[3a,6-dimethyl-5,7-dioxo-(3'R,3aS,6R)-dis...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067819(3-[3a,6-dimethyl-5,7-dioxo-(3'R,3aS,6R)-dispiro[pe...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067847(4-[(3aR,6R,9S)-6-(2-Carboxy-ethyl)-3a,6,9-trimethy...)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067821(4''-(1,3-dioxolan-2-yl)-2'',15''-dimethyl-(2''R,5'...)
Affinity DataIC50: 3.80E+4nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067823(Isobutyric acid 2-[(3aS,6R)-6-(2-carboxy-ethyl)-3a...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067827((S)-2-[(3aR,6R,9S)-3-(1,5-Dimethyl-hexyl)-9-ethyl-...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067826(3-[(3aR,6R)-3-(1,5-Dimethyl-hexyl)-3a,6-dimethyl-7...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067844(2-((10S,13S,17R)-17-hydroxy-10,13,16-trimethyl-3-o...)
Affinity DataIC50: 4.00E+4nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067818(3,3-Dimethyl-pentanedioic acid mono-[2-((9R,10S,11...)
Affinity DataIC50: 4.80E+4nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067828(3-Carboxy-pentanedioic acid mono-[2-((10R,13S,17R)...)
Affinity DataIC50: 5.00E+4nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067853(2-Ethyl-butyric acid 2-((10R,13S,17R)-17-hydroxy-1...)
Affinity DataIC50: 5.60E+4nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067820(3-[(3aR,6R,9S)-3-(1,5-Dimethyl-hexyl)-9-ethyl-3a,6...)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067838(2'',13'',15''-trimethyl-(2''R,5'R,13''S,15''S)-dis...)
Affinity DataIC50: 9.60E+4nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067845((7S,10R,13R)-17-(1,5-Dimethyl-hexyl)-7-ethyl-10,13...)
Affinity DataIC50: 1.00E+5nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067829(2'',13'',15''-trimethyl-(2''R,5'R,13''R,15''S)-dis...)
Affinity DataIC50: 1.00E+5nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067839((10R,13S)-17-(2-Hydroxy-acetyl)-10,13-dimethyl-1,6...)
Affinity DataIC50: 1.00E+5nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067840(3-[(3aR,6R,9S)-3-(1,5-Dimethyl-hexyl)-3a,6,9-trime...)
Affinity DataIC50: 1.00E+5nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067824(3-((3aS,6R)-3-Acetyl-3a,6-dimethyl-5,7-dioxo-dodec...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067850([(2S,10R,13R)-17-(1,5-Dimethyl-hexyl)-10,13-dimeth...)
Affinity DataIC50: 1.00E+5nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067822([(2S,10R,13R)-17-(1,5-Dimethyl-hexyl)-10,13-dimeth...)
Affinity DataIC50: 1.00E+5nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067837(2-Ethyl-butyric acid 2-((10R,11S,13S,17R)-11,17-di...)
Affinity DataIC50: 1.00E+5nMAssay Description:inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067832(3a,6-dimethyl-5,7-dioxo-(3'R,3aS,6R)-dispiro[perhy...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
LigandPNGBDBM50067836((S)-2-[(3aR,6R)-3-(1,5-Dimethyl-hexyl)-3a,6-dimeth...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed