Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50034929
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50069673(6-Nitro-7-(4-phenyl-piperidin-1-ylmethyl)-1,4-dihy...)
Affinity DataIC50: 330nMAssay Description:Tested for in vitro binding affinity against glycine-bining site of NMDA receptor using [3H]MDL-105519 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50069692(1-(7-Nitro-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 590nMAssay Description:Tested for in vitro binding affinity against glycine-bining site of NMDA receptor using [3H]MDL-105519 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50069684(1-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 840nMAssay Description:Tested for in vitro binding affinity against glycine-bining site of NMDA receptor using [3H]MDL-105519 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50069668(6-Azetidin-1-ylmethyl-7-nitro-1,4-dihydro-quinoxal...)
Affinity DataIC50: 3.80E+3nMAssay Description:Tested for in vitro binding affinity against glycine-bining site of NMDA receptor using [3H]MDL-105519 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50069690(1-(7-Nitro-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 3.90E+3nMAssay Description:Tested for in vitro binding affinity against glycine-bining site of NMDA receptor using [3H]MDL-105519 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed