Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50008014
LigandPNGBDBM50070088(3-{1-[2-(2-Hydroxy-ethoxy)-ethyl]-1H-indol-3-yl}-4...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory concentration was determined by measuring phosphorylation of H1 histone using active human Cell division cycle 2-cyclin B complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50070093(3,4-bis(indol-3-yl)maleimide derivative | CHEMBL73...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibitory concentration was determined by measuring phosphorylation of H1 histone using active human Cell division cycle 2-cyclin B complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM2583(bis-indolylmaleimide deriv. 8a | 3,4-bis(1H-indol-...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibitory concentration was determined by measuring phosphorylation of H1 histone using active human Cell division cycle 2-cyclin B complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM2683(2-[1-(3-dimethylaminopropyl)-indol-3-yl]-3-(indol-...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibitory concentration was determined by measuring phosphorylation of H1 histone using active human Cell division cycle 2-cyclin B complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50070082(3-[1-(3-Dimethylamino-propyl)-1H-indol-3-yl]-4-{1-...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibitory concentration was determined by measuring phosphorylation of H1 histone using active human Cell division cycle 2-cyclin B complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50070084(3,4-bis(indol-3-yl)maleimide derivative | CHEMBL38...)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibitory concentration was determined by measuring phosphorylation of H1 histone using active human Cell division cycle 2-cyclin B complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50070090(3-[1-(3-Dimethylamino-propyl)-1H-indol-3-yl]-4-(1-...)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibitory concentration was determined by measuring phosphorylation of H1 histone using active human Cell division cycle 2-cyclin B complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50070092(3-[1-(2-{2-[2-(2-Hydroxy-ethoxy)-ethoxy]-ethoxy}-e...)
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibitory concentration was determined by measuring phosphorylation of H1 histone using active human Cell division cycle 2-cyclin B complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50070087((S)-1-{(R)-2-Acetylamino-3-[2-(2-{3-[4-(1H-indol-3...)
Affinity DataIC50: 9.80E+4nMAssay Description:Inhibitory concentration was determined by measuring phosphorylation of H1 histone using active human Cell division cycle 2-cyclin B complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50070086(3,4-bis(indol-3-yl)maleimide derivative | CHEMBL43...)
Affinity DataIC50: 2.20E+5nMAssay Description:Inhibitory concentration was determined by measuring phosphorylation of H1 histone using active human Cell division cycle 2-cyclin B complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50070089(3-(1-{2-[2-(2-Hydroxy-ethoxy)-ethoxy]-ethyl}-1H-in...)
Affinity DataIC50: 2.85E+5nMAssay Description:Inhibitory concentration was determined by measuring phosphorylation of H1 histone using active human Cell division cycle 2-cyclin B complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50070085(3,4-bis(indol-3-yl)maleimide derivative | CHEMBL38...)
Affinity DataIC50: 5.70E+5nMAssay Description:Inhibitory concentration was determined by measuring phosphorylation of H1 histone using active human Cell division cycle 2-cyclin B complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50070091(3,4-bis(indol-3-yl)maleimide derivative | CHEMBL42...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory concentration was determined by measuring phosphorylation of H1 histone using active human Cell division cycle 2-cyclin B complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50070094((S)-1-((R)-2-Acetylamino-3-mercapto-propionyl)-pyr...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory concentration was determined by measuring phosphorylation of H1 histone using active human Cell division cycle 2-cyclin B complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50070083(3,4-bis(indol-3-yl)maleimide derivative | CHEMBL42...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory concentration was determined by measuring phosphorylation of H1 histone using active human Cell division cycle 2-cyclin B complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed