Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50008016
TargetAromatase(Human)
Centre D'Etudes Et De Recherche Sur Le MéDicament De Normandie

Curated by ChEMBL
LigandPNGBDBM8611(CHEMBL468419 | 4-{5H,6H,7H,8H-imidazo[1,5-a]pyridi...)
Affinity DataKi:  0.600nMAssay Description:Inhibition constant for human aromatase cytochrome P450 19A1 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Centre D'Etudes Et De Recherche Sur Le MéDicament De Normandie

Curated by ChEMBL
LigandPNGBDBM50070095(3-Phenyl-2-[1-pyridin-4-yl-meth-(Z)-ylidene]-indan...)
Affinity DataKi:  10nMAssay Description:Inhibition constant for human aromatase cytochrome P450 19A1 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Centre D'Etudes Et De Recherche Sur Le MéDicament De Normandie

Curated by ChEMBL
LigandPNGBDBM50070097(MR-20492 | (Z)-6-(4-chlorophenyl)-7-(pyridin-4-ylm...)
Affinity DataKi:  10nMAssay Description:Inhibition constant for human aromatase cytochrome P450 19A1 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Centre D'Etudes Et De Recherche Sur Le MéDicament De Normandie

Curated by ChEMBL
LigandPNGBDBM50215414(MR-20814 | CHEMBL1096024)
Affinity DataKi:  86nMAssay Description:Inhibition constant for human aromatase cytochrome P450 19A1 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Centre D'Etudes Et De Recherche Sur Le MéDicament De Normandie

Curated by ChEMBL
LigandPNGBDBM50070097(MR-20492 | (Z)-6-(4-chlorophenyl)-7-(pyridin-4-ylm...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human aromatase cytochrome P450 19A1 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Centre D'Etudes Et De Recherche Sur Le MéDicament De Normandie

Curated by ChEMBL
LigandPNGBDBM8611(CHEMBL468419 | 4-{5H,6H,7H,8H-imidazo[1,5-a]pyridi...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human aromatase cytochrome P450 19A1 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Centre D'Etudes Et De Recherche Sur Le MéDicament De Normandie

Curated by ChEMBL
LigandPNGBDBM50070095(3-Phenyl-2-[1-pyridin-4-yl-meth-(Z)-ylidene]-indan...)
Affinity DataIC50: 800nMAssay Description:Inhibition of human aromatase cytochrome P450 19A1 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Centre D'Etudes Et De Recherche Sur Le MéDicament De Normandie

Curated by ChEMBL
LigandPNGBDBM50215414(MR-20814 | CHEMBL1096024)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human aromatase cytochrome P450 19A1 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed