Report error Found 94 Enz. Inhib. hit(s) with all data for entry = 50008023
Affinity DataEC50: <0.100nMAssay Description:Compound was tested for agonist activity against cloned human beta-2 adrenergic receptor at a concentration of 1000 nMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.770nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Agonist activity against cloned human beta-1 adrenergic receptor as percent activation of adenyl cyclase activity at a concentration of 1000 nMMore data for this Ligand-Target Pair
Affinity DataEC50: 4.30nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 4.80nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Compound was tested for agonist activity against cloned human beta-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 5.40nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 5.90nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70nMAssay Description:Agonist activity against cloned human beta-1 adrenergic receptor as percent activation of adenyl cyclase activity at a concentration of 1000 nMMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Compound was tested for binding affinity against cloned human beta-1 adrenergic receptor from CHO cells using [125I]-iodocyanopindolol as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Binding affinity against cloned human beta-2 adrenergic receptor from CHO cells using [125I]iodocyanopindolol as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Binding affinity against cloned human beta-2 adrenergic receptor from CHO cells using [125I]iodocyanopindolol as the radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Compound was tested for agonist activity against cloned human beta-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Agonist activity against cloned human beta-1 adrenergic receptor as percent activation of adenyl cyclase activity at a concentration of 1000 nMMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Binding affinity against cloned human beta-2 adrenergic receptor from CHO cells using [125I]iodocyanopindolol as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Binding affinity against cloned human beta-2 adrenergic receptor from CHO cells using [125I]iodocyanopindolol as the radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Agonist activity against cloned human beta-1 adrenergic receptor as percent activation of adenyl cyclase activity at a concentration of 1000 nMMore data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Compound was tested for agonist activity against cloned human beta-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 39nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 54nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 58nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Binding affinity against cloned human beta-2 adrenergic receptor from CHO cells using [125I]iodocyanopindolol as the radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Agonist activity against cloned human beta-1 adrenergic receptor as percent activation of adenyl cyclase activity at a concentration of 1000 nMMore data for this Ligand-Target Pair
Affinity DataEC50: 62nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Binding affinity against cloned human beta-2 adrenergic receptor from CHO cells using [125I]iodocyanopindolol as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Agonist activity against cloned human beta-1 adrenergic receptor as percent activation of adenyl cyclase activity at a concentration of 1000 nMMore data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Binding affinity against cloned human beta-2 adrenergic receptor from CHO cells using [125I]iodocyanopindolol as the radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 92nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Agonist activity against cloned human beta-1 adrenergic receptor as percent activation of adenyl cyclase activity at a concentration of 1000 nMMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Binding affinity against cloned human beta-2 adrenergic receptor from CHO cells using [125I]iodocyanopindolol as the radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Agonist activity against cloned human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Agonist activity against cloned human beta-1 adrenergic receptor as percent activation of adenyl cyclase activity at a concentration of 1000 nMMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Binding affinity against cloned human beta-2 adrenergic receptor from CHO cells using [125I]iodocyanopindolol as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Binding affinity against cloned human beta-2 adrenergic receptor from CHO cells using [125I]iodocyanopindolol as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Binding affinity against cloned human beta-2 adrenergic receptor from CHO cells using [125I]iodocyanopindolol as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Tested for binding affinity against cloned human beta-1 adrenergic receptor from CHO cells using [125I]iodocyanopindolol as the radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Tested for binding affinity against cloned human beta-1 adrenergic receptor from CHO cells using [125I]iodocyanopindolol as the radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Binding affinity against cloned human beta-2 adrenergic receptor from CHO cells using [125I]iodocyanopindolol as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Agonist activity against cloned human beta-1 adrenergic receptor as percent activation of adenyl cyclase activity at a concentration of 1000 nMMore data for this Ligand-Target Pair


























