Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50008153
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50403654(CHEMBL2115073)
Affinity DataKi:  0.840nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071118(CHEMBL2111522 | N-[2-(3,4-Dichloro-phenyl)-4-(4-{1...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071112(SR 48968 | CHEMBL56835 | N-[4-(4-Acetylamino-4-phe...)
Affinity DataKi:  1.75nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071112(SR 48968 | CHEMBL56835 | N-[4-(4-Acetylamino-4-phe...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216091(CHEMBL2111522)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071118(CHEMBL2111522 | N-[2-(3,4-Dichloro-phenyl)-4-(4-{1...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071125(N-{2-(3,4-Dichloro-phenyl)-4-[4-(1-ethyl-1-hydroxy...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071120(N-{2-(3,4-Dichloro-phenyl)-4-[4-(1-hydroxy-butyl)-...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071119(N-{2-(3,4-Dichloro-phenyl)-4-[4-(1-hydroxy-1-propy...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071115(N-[2-(3,4-Dichloro-phenyl)-4-(4-{1-[(E)-methoxyimi...)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071121(N-{2-(3,4-Dichloro-phenyl)-4-[4-(1-hydroxy-1-methy...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071122(N-[2-(3,4-Dichloro-phenyl)-4-(4-propionyl-piperidi...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071126(N-[2-(3,4-Dichloro-phenyl)-4-(4-propyl-piperidin-1...)
Affinity DataKi:  9.90nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071124(N-{2-(3,4-Dichloro-phenyl)-4-[4-(1-hydroxy-propyl)...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071123(N-{2-(3,4-Dichloro-phenyl)-4-[4-(1-hydroxy-ethyl)-...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071113(Acetic acid 2-{1-[4-(benzoyl-methyl-amino)-3-(3,4-...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071117(N-{2-(3,4-Dichloro-phenyl)-4-[4-(2-hydroxy-ethyl)-...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071116(N-[4-[4-(2-Acetylamino-ethyl)-piperidin-1-yl]-2-(3...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071114(N-[2-(3,4-Dichloro-phenyl)-4-(4-hydroxymethyl-pipe...)
Affinity DataKi:  142nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed