Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50008200
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071445(N-[(R)-1-[(S)-2-Ethenesulfonylamino-1-(1H-indol-3-...)
Affinity DataKi:  0.140nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071438((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  0.210nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071435((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071437(N-[(R)-1-[(S)-1-(1H-Indol-3-ylmethyl)-2-oxo-2-(pro...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071423(N-[(R)-1-[(S)-2-(2-Ethoxy-ethanesulfonylamino)-1-(...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071420(N-[(R)-1-[(S)-1-(1H-Indol-3-ylmethyl)-2-oxo-2-(pro...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071436(N-[(R)-1-[(S)-2-(Butane-1-sulfonylamino)-1-(1H-ind...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071421(N-[(R)-1-[(S)-2-Benzenesulfonylamino-1-(1H-indol-3...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071439(N-[(R)-1-[(S)-1-(1H-Indol-3-ylmethyl)-2-oxo-2-(pro...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071430(N-[(R)-1-[(S)-2-Ethanesulfonylamino-1-(1H-indol-3-...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071428(N-[(R)-1-{(S)-1-(1H-Indol-3-ylmethyl)-2-oxo-2-[((E...)
Affinity DataKi:  0.390nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071444(N-[(R)-1-[1-(Butane-1-sulfonylaminocarbonyl)-3-met...)
Affinity DataKi:  0.490nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071443(N-[(R)-1-[(S)-1-(1H-Indol-3-ylmethyl)-2-oxo-2-phen...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071440(N-[(R)-1-[2-(Butane-1-sulfonylamino)-1-naphthalen-...)
Affinity DataKi:  0.590nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071432((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071426(N-[(R)-1-[1-(Butane-1-sulfonylaminocarbonyl)-propy...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071441((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  0.760nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071427((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  0.790nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071437(N-[(R)-1-[(S)-1-(1H-Indol-3-ylmethyl)-2-oxo-2-(pro...)
Affinity DataKi:  0.890nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071433((S)-2-{(R)-3-Biphenyl-4-yl-2-[(3,5-dimethyl-benzoy...)
Affinity DataKi:  1nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071425(N-[(R)-1-[(S)-1-(Butane-1-sulfonylaminocarbonyl)-2...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071434(N-[(R)-1-[1-(Butane-1-sulfonylaminocarbonyl)-3-met...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071425(N-[(R)-1-[(S)-1-(Butane-1-sulfonylaminocarbonyl)-2...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071445(N-[(R)-1-[(S)-2-Ethenesulfonylamino-1-(1H-indol-3-...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071420(N-[(R)-1-[(S)-1-(1H-Indol-3-ylmethyl)-2-oxo-2-(pro...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071421(N-[(R)-1-[(S)-2-Benzenesulfonylamino-1-(1H-indol-3...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071436(N-[(R)-1-[(S)-2-(Butane-1-sulfonylamino)-1-(1H-ind...)
Affinity DataKi:  2.90nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071442(N-[(R)-1-[2-(Butane-1-sulfonylamino)-1-cyclohexyl-...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071440(N-[(R)-1-[2-(Butane-1-sulfonylamino)-1-naphthalen-...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071424(N-[(R)-1-[1-(Butane-1-sulfonylaminocarbonyl)-2-hyd...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071422(N-[(R)-1-[1-(Butane-1-sulfonylaminocarbonyl)-2-met...)
Affinity DataKi:  3.5nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071428(N-[(R)-1-{(S)-1-(1H-Indol-3-ylmethyl)-2-oxo-2-[((E...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071429((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071444(N-[(R)-1-[1-(Butane-1-sulfonylaminocarbonyl)-3-met...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071430(N-[(R)-1-[(S)-2-Ethanesulfonylamino-1-(1H-indol-3-...)
Affinity DataKi:  5.30nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071443(N-[(R)-1-[(S)-1-(1H-Indol-3-ylmethyl)-2-oxo-2-phen...)
Affinity DataKi:  5.40nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071426(N-[(R)-1-[1-(Butane-1-sulfonylaminocarbonyl)-propy...)
Affinity DataKi:  5.5nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071423(N-[(R)-1-[(S)-2-(2-Ethoxy-ethanesulfonylamino)-1-(...)
Affinity DataKi:  6nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071422(N-[(R)-1-[1-(Butane-1-sulfonylaminocarbonyl)-2-met...)
Affinity DataKi:  6.90nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071434(N-[(R)-1-[1-(Butane-1-sulfonylaminocarbonyl)-3-met...)
Affinity DataKi:  8nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071442(N-[(R)-1-[2-(Butane-1-sulfonylamino)-1-cyclohexyl-...)
Affinity DataKi:  8.60nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071424(N-[(R)-1-[1-(Butane-1-sulfonylaminocarbonyl)-2-hyd...)
Affinity DataKi:  9.10nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071439(N-[(R)-1-[(S)-1-(1H-Indol-3-ylmethyl)-2-oxo-2-(pro...)
Affinity DataKi:  10nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071431((S)-2-{(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  36nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071438((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  45nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071435((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  54nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071432((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  87nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071427((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  130nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071441((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  250nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Takarazuka Research Institute

Curated by ChEMBL
LigandPNGBDBM50071433((S)-2-{(R)-3-Biphenyl-4-yl-2-[(3,5-dimethyl-benzoy...)
Affinity DataKi:  440nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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