Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50008371
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50072753((S)-1-[(3S,4R)-3-(Benzo[1,3]dioxol-5-yloxymethyl)-...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50072748(1-{6-[(3R,4S)-3-(Benzo[1,3]dioxol-5-yloxymethyl)-4...)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50072745((S)-1-(1H-Indol-4-yloxy)-3-[(S)-3-phenyl-3-(4-trif...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50072743((R)-1-[(3S,4R)-3-(Benzo[1,3]dioxol-5-yloxymethyl)-...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50072752(1-(1H-Indol-4-yloxy)-3-[3-phenyl-3-(4-trifluoromet...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50072746((S)-1-(Naphthalen-1-yloxy)-3-[(S)-3-phenyl-3-(4-tr...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50072751(1-(2-Cyclopentyl-phenoxy)-3-[3-phenyl-3-(4-trifluo...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50072754((1S,2R)-2-{[2-Hydroxy-3-(1H-indol-4-yloxy)-propyla...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50072750((R)-1-(1H-Indol-4-yloxy)-3-[(S)-3-phenyl-3-(4-trif...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50072755((2S)-1-(1H-indol-4-yloxy)-3-[(propan-2-yl)amino]pr...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50072744((R)-1-(Naphthalen-1-yloxy)-3-[(S)-3-phenyl-3-(4-tr...)
Affinity DataKi:  142nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50072747(1-{6-[(3R,4S)-3-(Benzo[1,3]dioxol-5-yloxymethyl)-4...)
Affinity DataKi:  156nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50072749(1-(Naphthalen-1-yloxy)-3-{6-[3-phenyl-3-(4-trifluo...)
Affinity DataKi:  391nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed