Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50008469
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataIC50: 0.0600nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50033857(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50033852(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50: 0.540nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50033839(1-(2-Methoxy-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50: 0.770nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073621(1-(2-Methoxy-phenyl)-4-[3-((S)-5-methoxy-1,2,3,4-t...)
Affinity DataIC50: 1.30nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073614(1-(2-Methoxy-phenyl)-4-[3-((R)-5-methoxy-1,2,3,4-t...)
Affinity DataIC50: 1.60nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073617(1-[3-((S)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50: 2.30nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073620(1-[3-((S)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50: 2.40nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073622(7,7-Bis-(3-amino-propyl)-5,6,7,8-tetrahydro-naphth...)
Affinity DataIC50: 2.5nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073610(1-[3-((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50: 4.30nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073613(1-[3-((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50: 4.5nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073615({2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-((...)
Affinity DataIC50: 7nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073619({3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-(...)
Affinity DataIC50: 7nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50033847({2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-(5...)
Affinity DataIC50: 7.70nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073612({2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-((...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50052569({3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-(...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50033839(1-(2-Methoxy-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50: 18nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073611({3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-(...)
Affinity DataIC50: 34nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073621(1-(2-Methoxy-phenyl)-4-[3-((S)-5-methoxy-1,2,3,4-t...)
Affinity DataIC50: 38nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50052563(N-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-3-...)
Affinity DataIC50: 38nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataIC50: 50nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073616(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-((S)-5-m...)
Affinity DataIC50: 89nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50033857(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50: 110nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50033852(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50: 140nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073614(1-(2-Methoxy-phenyl)-4-[3-((R)-5-methoxy-1,2,3,4-t...)
Affinity DataIC50: 150nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073618(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-((R)-5-m...)
Affinity DataIC50: 320nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50033847({2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-(5...)
Affinity DataIC50: 380nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073617(1-[3-((S)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50: 600nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073620(1-[3-((S)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50: 610nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073615({2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-((...)
Affinity DataIC50: 650nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50052563(N-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-3-...)
Affinity DataIC50: 761nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073618(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-((R)-5-m...)
Affinity DataIC50: 870nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073613(1-[3-((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50: 880nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073610(1-[3-((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50: 880nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50052569({3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-(...)
Affinity DataIC50: 1.06E+3nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073619({3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-(...)
Affinity DataIC50: 1.90E+3nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073611({3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}-(...)
Affinity DataIC50: 2.30E+3nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073616(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-((S)-5-m...)
Affinity DataIC50: 2.60E+3nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50073612({2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-((...)
Affinity DataIC50: 3.20E+3nMAssay Description:In vitro inhibition of [3H]spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed