Compile Data Set for Download or QSAR
Report error Found 117 Enz. Inhib. hit(s) with all data for entry = 637
LigandPNGBDBM284822(US10023576, Example 12 | 1-((cis)-4-(5-(4-amino-5-...)
Affinity DataIC50: 0.400nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284900(US10023576, Example 91 | (S)-4-acetyl-1-(5-(4-amin...)
Affinity DataIC50: 0.550nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284821(US10023576, Example 11 | 1-((cis)-4-(5-(4-amino-5-...)
Affinity DataIC50: 0.600nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284825(US10023576, Example 15 | 1-(4-(5-(4-amino-5-(1-(te...)
Affinity DataIC50: 0.600nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284823(US10023576, Example 13 | 1-((cis)-4-(5-(4-amino-5-...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284824(US10023576, Example 14 | 1-(4-(5-(4-amino-5-(1-(te...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284826(US10023576, Example 16 | 7-(1-(Tetrahydro-2H-pyran...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284831(US10023576, Example 21 | 1-(4-(6-(4-amino-5-(1-(te...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284842(US10023576, Example 32 | 5-(1-cyclohexyl-1H-1,2,3-...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284856(US10023576, Example 46 | 7-(1-(cyclopropylmethyl)-...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284872(US10023576, Example 63 | 7-(2-(4-(oxetan-3-yl)pipe...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284893(US10023576, Example 84 | 4-acetyl-1-(5-(4-amino-5-...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284899(US10023576, Example 90 | (R)-1-(4-(4-amino-5-(1-(1...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284901(US10023576, Example 92 | (S)-4-acetyl-1-(5-(4-amin...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284902(US10023576, Example 93 | (S)-4-acetyl-1-(4-(4-amin...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284906(US10023576, Example 98 | (S)-4-acetyl-1-(4-(4-amin...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284910(US10023576, Example 102 | (S)-4-acetyl-1-(5-(4-ami...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284912(US10023576, Example 104 | ((S)-4-acetyl-1-(5-(4-am...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284818(US10023576, Example 8 | 4-(5-(4-amino-5-(1-isoprop...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284819(US10023576, Example 9 | 1-((cis)-4-(5-(4-amino-5-(...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284828(US10023576, Example 18 | 5-(6-(4-Amino-5-(1-(tetra...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284830(US10023576, Example 20 | 1-(4-(6-(4-amino-5-(1-(te...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284834(US10023576, Example 24 | 5-(1-(tetrahydro-2H-pyran...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284835(US10023576, Example 25 | 5-(1-isopropyl-1H-1,2,3-t...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284837(US10023576, Example 27 | 7-(1-(2,6-dimethyltetrahy...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
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LigandPNGBDBM284838(US10023576, Example 28 | 7-(3-methyl-1-(tetrahydro...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284839(US10023576, Example 29 | 7-(3-methyl-1-(tetrahydro...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284840(US10023576, Example 30 | 7-(1-(tetrahydro-2H-pyran...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284841(US10023576, Example 31 | 5-(1-(tetrahydro-2H-pyran...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284843(US10023576, Example 33 | 4-(6-(4-amino-5-(1-(tetra...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284846(US10023576, Example 36 | 4-(6-(4-amino-5-(1-(tetra...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284849(US10023576, Example 39 | 4-(6-(4-amino-5-(1-(tetra...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284855(US10023576, Example 45 | 7-(1-(cyclopropylmethyl)-...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284864(US10023576, Example 55 | 2-(6-(4-amino-5-(1-(tetra...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284871(US10023576, Example 62 | 7-(2-(piperazin-1-yl)pyri...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284864(US10023576, Example 55 | 2-(6-(4-amino-5-(1-(tetra...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284890(US10023576, Example 81 | 2-(6-(4-amino-5-(1-(tetra...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284895(US10023576, Example 86 | 1-(5-(4-amino-5-chloropyr...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284897(US10023576, Example 88 | 4-acetyl-1-(5-(4-amino-5-...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284898(US10023576, Example 89 | 1-(5-(4-amino-5-(1-(tetra...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284907(US10023576, Example 99 | (S)-4-(5-(4-amino-5-(trif...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284909(US10023576, Example 101 | (R)-4-(5-(4-amino-5-(tri...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284917(US10023576, Example 109 | (S)-7-(6-(4-acetyl-3,3,6...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284919(US10023576, Example 111 | (S)-4-acetyl-1-(6-(4-ami...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284850(US10023576, Example 40 | 4-(6-(4-amino-5-(1-(tetra...)
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284857(US10023576, Example 47 | 7-(1-((2,2-difluorocyclop...)
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284858(US10023576, Example 48 | 7-(1-((2,2-difluorocyclop...)
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284875(US10023576, Example 66 | 2-(4-(4-Amino-5-(1-(tetra...)
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284876(US10023576, Example 67 | 2-(5-(4-Amino-5-(1-(tetra...)
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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LigandPNGBDBM284878(US10023576, Example 69 | 7-[1-(oxan-4-yl)-1H-indaz...)
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:The ADP-Glo format PI3K assays were performed in Proxiplate 384-well plates (Perkin Elmer #6008280). The final assay volume was 2 μl prepared fr...More data for this Ligand-Target Pair
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Date in BDB:
1/11/2019
Entry Details
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