Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 899
TargetGag-Pol polyprotein(HIV-1)
Viiv Healthcare

US Patent
LigandPNGBDBM297496(US10118894, Example 5)
Affinity DataIC50: 5nMAssay Description:Antiviral HIV activity and cytotoxicity values for compounds of the invention from Table 1 were measured in parallel in the HTLV-1 transformed cell l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Viiv Healthcare

US Patent
LigandPNGBDBM297498(US10118894, Example 7)
Affinity DataIC50: 14nMAssay Description:Antiviral HIV activity and cytotoxicity values for compounds of the invention from Table 1 were measured in parallel in the HTLV-1 transformed cell l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Viiv Healthcare

US Patent
LigandPNGBDBM297492(US10118894, Example 1)
Affinity DataIC50: 25nMAssay Description:Antiviral HIV activity and cytotoxicity values for compounds of the invention from Table 1 were measured in parallel in the HTLV-1 transformed cell l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Viiv Healthcare

US Patent
LigandPNGBDBM297497(US10118894, Example 6)
Affinity DataIC50: 36nMAssay Description:Antiviral HIV activity and cytotoxicity values for compounds of the invention from Table 1 were measured in parallel in the HTLV-1 transformed cell l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Viiv Healthcare

US Patent
LigandPNGBDBM297493(US10118894, Example 2)
Affinity DataIC50: 42nMAssay Description:Antiviral HIV activity and cytotoxicity values for compounds of the invention from Table 1 were measured in parallel in the HTLV-1 transformed cell l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Viiv Healthcare

US Patent
LigandPNGBDBM297495(US10118894, Example 4)
Affinity DataIC50: 52nMAssay Description:Antiviral HIV activity and cytotoxicity values for compounds of the invention from Table 1 were measured in parallel in the HTLV-1 transformed cell l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Viiv Healthcare

US Patent
LigandPNGBDBM297494(US10118894, Example 3)
Affinity DataIC50: 86nMAssay Description:Antiviral HIV activity and cytotoxicity values for compounds of the invention from Table 1 were measured in parallel in the HTLV-1 transformed cell l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
Go to US Patent