Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 2481
TargetCannabinoid receptor 1(Rat)
Uti Limited Partnership

US Patent
LigandPNGBDBM368196(US10227332, No. 10)
Affinity DataKi:  15nMAssay Description:The structure-activity relationship and optimization studies have led to the discovery of selective T-type calcium channel blockers, e.g., compound 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
US Patent

TargetCannabinoid receptor 1(Rat)
Uti Limited Partnership

US Patent
LigandPNGBDBM368194(US10227332, No. 8)
Affinity DataKi:  283nMAssay Description:The structure-activity relationship and optimization studies have led to the discovery of selective T-type calcium channel blockers, e.g., compound 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
US Patent

TargetCannabinoid receptor 2(Human)
Uti Limited Partnership

US Patent
LigandPNGBDBM368196(US10227332, No. 10)
Affinity DataKi:  1.97E+3nMAssay Description:The structure-activity relationship and optimization studies have led to the discovery of selective T-type calcium channel blockers, e.g., compound 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
US Patent

TargetCannabinoid receptor 2(Human)
Uti Limited Partnership

US Patent
LigandPNGBDBM368194(US10227332, No. 8)
Affinity DataKi:  2.83E+3nMAssay Description:The structure-activity relationship and optimization studies have led to the discovery of selective T-type calcium channel blockers, e.g., compound 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
US Patent

TargetCannabinoid receptor 2(Human)
Uti Limited Partnership

US Patent
LigandPNGBDBM368193(US10227332, No. 6)
Affinity DataKi:  2.96E+3nMAssay Description:The structure-activity relationship and optimization studies have led to the discovery of selective T-type calcium channel blockers, e.g., compound 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
US Patent

TargetCannabinoid receptor 1(Rat)
Uti Limited Partnership

US Patent
LigandPNGBDBM368193(US10227332, No. 6)
Affinity DataKi: >5.00E+3nMAssay Description:The structure-activity relationship and optimization studies have led to the discovery of selective T-type calcium channel blockers, e.g., compound 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
US Patent

TargetCannabinoid receptor 2(Human)
Uti Limited Partnership

US Patent
LigandPNGBDBM368195(US10227332, No. 9)
Affinity DataKi: >5.00E+3nMAssay Description:The structure-activity relationship and optimization studies have led to the discovery of selective T-type calcium channel blockers, e.g., compound 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
US Patent

TargetCannabinoid receptor 1(Rat)
Uti Limited Partnership

US Patent
LigandPNGBDBM368195(US10227332, No. 9)
Affinity DataKi: >5.00E+3nMAssay Description:The structure-activity relationship and optimization studies have led to the discovery of selective T-type calcium channel blockers, e.g., compound 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
US Patent