Compile Data Set for Download or QSAR
Report error Found 80 Enz. Inhib. hit(s) with all data for entry = 2988
TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387751(US10294214, Example 51)
Affinity DataEC50:  1.00E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387760(US10294214, Example 60)
Affinity DataEC50:  200nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387759(US10294214, Example 59)
Affinity DataEC50:  200nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387758(US10294214, Example 58)
Affinity DataEC50:  79.4nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387757(US10294214, Example 57)
Affinity DataEC50:  2.51E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387756(US10294214, Example 56)
Affinity DataEC50:  1.26E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387755(US10294214, Example 55)
Affinity DataEC50:  1.59E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387754(US10294214, Example 54)
Affinity DataEC50:  1.00E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387753(US10294214, Example 53)
Affinity DataEC50:  2.00E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387752(US10294214, Example 52)
Affinity DataEC50:  1.26E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387761(US10294214, Example 61)
Affinity DataEC50:  251nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387750(US10294214, Example 50)
Affinity DataEC50:  794nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387749(US10294214, Example 49)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387748(US10294214, Example 48)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387747(US10294214, Example 47)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387746(US10294214, Example 46)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387745(US10294214, Example 45)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387744(US10294214, Example 44)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387743(US10294214, Example 43)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387742(US10294214, Example 42)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387771(US10294214, Example 71)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387780(US10294214, Example 80)
Affinity DataEC50:  1.00E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387779(US10294214, Example 79)
Affinity DataEC50:  794nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387778(US10294214, Example 78)
Affinity DataEC50:  1.00E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387777(US10294214, Example 77)
Affinity DataEC50:  1.59E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387776(US10294214, Example 76)
Affinity DataEC50:  2.00E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387775(US10294214, Example 75)
Affinity DataEC50:  1.26E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387774(US10294214, Example 74)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387773(US10294214, Example 73)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387772(US10294214, Example 72)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387741(US10294214, Example 41)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387770(US10294214, Example 70)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387769(US10294214, Example 69)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387768(US10294214, Example 68)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387767(US10294214, Example 67)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387766(US10294214, Example 66)
Affinity DataEC50:  251nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387765(US10294214, Example 65)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387764(US10294214, Example 64)
Affinity DataEC50:  251nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387763(US10294214, Example 63)
Affinity DataEC50:  200nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387762(US10294214, Example 62)
Affinity DataEC50:  251nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387711(US10294214, Example 11)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387720(US10294214, Example 20)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387719(US10294214, Example 19)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387718(US10294214, Example 18)
Affinity DataEC50:  794nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387717(US10294214, Example 17)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387716(US10294214, Example 16)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387715(US10294214, Example 15)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387714(US10294214, Example 14)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387713(US10294214, Example 13)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387712(US10294214, Example 12)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent

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