Compile Data Set for Download or QSAR
Report error Found 80 Enz. Inhib. hit(s) with all data for entry = 2988
TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387758(US10294214, Example 58)
Affinity DataEC50:  79.4nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387703(methyl 3-(2-(4-cyclohexylpiperidin-1-yl)acetamido)...)
Affinity DataEC50:  200nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387759(US10294214, Example 59)
Affinity DataEC50:  200nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387763(US10294214, Example 63)
Affinity DataEC50:  200nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387760(US10294214, Example 60)
Affinity DataEC50:  200nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387766(US10294214, Example 66)
Affinity DataEC50:  251nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387764(US10294214, Example 64)
Affinity DataEC50:  251nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387739(US10294214, Example 39)
Affinity DataEC50:  251nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387738(US10294214, Example 38)
Affinity DataEC50:  251nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387737(US10294214, Example 37)
Affinity DataEC50:  251nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387762(US10294214, Example 62)
Affinity DataEC50:  251nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387761(US10294214, Example 61)
Affinity DataEC50:  251nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387767(US10294214, Example 67)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387765(US10294214, Example 65)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387705(US10294214, Example 5)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387704(US10294214, Example 4)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387711(US10294214, Example 11)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387742(US10294214, Example 42)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387710(US10294214, Example 10)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387740(US10294214, Example 40)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387708(US10294214, Example 8)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387771(US10294214, Example 71)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387707(US10294214, Example 7)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387770(US10294214, Example 70)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387706(US10294214, Example 6)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387768(US10294214, Example 68)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387743(US10294214, Example 43)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387741(US10294214, Example 41)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387709(US10294214, Example 9)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387744(US10294214, Example 44)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387702(N-(2-(cyclopropanecarbonyl)-1H-indol-3-yl)-2-(8-az...)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387748(US10294214, Example 48)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387769(US10294214, Example 69)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387772(US10294214, Example 72)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387746(US10294214, Example 46)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387745(US10294214, Example 45)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387713(US10294214, Example 13)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387712(US10294214, Example 12)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387719(US10294214, Example 19)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387749(US10294214, Example 49)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387717(US10294214, Example 17)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387716(US10294214, Example 16)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387722(US10294214, Example 22)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387721(US10294214, Example 21)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387720(US10294214, Example 20)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387774(US10294214, Example 74)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387773(US10294214, Example 73)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387747(US10294214, Example 47)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387715(US10294214, Example 15)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM387714(US10294214, Example 14)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
US Patent

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