Compile Data Set for Download or QSAR
Report error Found 69 Enz. Inhib. hit(s) with all data for entry = 3421
TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400216(US10328054, Example Compound 69)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400218(US10328054, Example Compound 58)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400219(US10328054, Example Compound 59)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400212(US10328054, Example Compound 65)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400213(US10328054, Example Compound 66)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400214(US10328054, Example Compound 67)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400215(US10328054, Example Compound 68)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400208(US10328054, Example Compound 55)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400209(US10328054, Example Compound 56)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400211(US10328054, Example Compound 64)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400204(US10328054, Example Compound 51)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400205(US10328054, Example Compound 52)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400206(US10328054, Example Compound 53)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400207(US10328054, Example Compound 54)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400228(US10328054, Example Compound 15)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400229(US10328054, Example Compound 39)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400224(US10328054, Example Compound 11)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400225(US10328054, Example Compound 12)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400226(US10328054, Example Compound 13)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400227(US10328054, Example Compound 14)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400220(US10328054, Example Compound 60)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400221(US10328054, Example Compound 7)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400222(US10328054, Example Compound 8)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400169(US10328054, Example Compound 20)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400164(US10328054, Example Compound 10)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400165(US10328054, Example Compound 16)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400166(US10328054, Example Compound 17)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400167(US10328054, Example Compound 18)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400161(US10328054, Example Compound 1 | Preparation of te...)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400162(US10328054, Example Compound 2 | Procedure for Pre...)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400184(US10328054, Example Compound 43)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400185(US10328054, Example Compound 50)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400186(US10328054, Example Compound 63)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400187(US10328054, Example Compound 5)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400180(US10328054, Example Compound 23)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400183(US10328054, Example Compound 38)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400176(US10328054, Example Compound 48)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400177(US10328054, Example Compound 62)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400178(US10328054, Example Compound 4 | Preparation of 1-...)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400179(US10328054, Example Compound 6)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400172(US10328054, Example Compound 40)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400173(US10328054, Example Compound 45)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400174(US10328054, Example Compound 46)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400175(US10328054, Example Compound 47)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400200(US10328054, Example Compound 41)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400201(US10328054, Example Compound 42)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400202(US10328054, Example Compound 44)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400203(US10328054, Example Compound 49)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400196(US10328054, Example Compound 34)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Hua Medicine (Shanghai)

US Patent
LigandPNGBDBM400197(US10328054, Example Compound 35)
Affinity DataIC50: 500nMAssay Description:For functional assays, HEK293 cells stably expressing recombinant rat mGluR5 were seeded in 384-well plates and dye loaded using Fluo-8. Cells were t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
US Patent

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