Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 8618
TargetDipeptidyl peptidase 4(Human)
Jiangsu Tasly Diyi Pharmaceutical

US Patent
LigandPNGBDBM408611(US10358449, Compound I-3)
Affinity DataIC50: 0.0800nMAssay Description:DPP-IV could hydrolyze Gly-Pro-Aminoluciferin at room temperature to generate Aminoluciferin, which could produce glow type luminescent signals in a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Jiangsu Tasly Diyi Pharmaceutical

US Patent
LigandPNGBDBM408607(US10358449, Compound I-1)
Affinity DataIC50: 0.210nMAssay Description:DPP-IV could hydrolyze Gly-Pro-Aminoluciferin at room temperature to generate Aminoluciferin, which could produce glow type luminescent signals in a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Jiangsu Tasly Diyi Pharmaceutical

US Patent
LigandPNGBDBM50228403(8-[(3R)-3-Aminopiperidin-1-yl]-7-but-2-yn-1-yl-3-m...)
Affinity DataIC50: 0.210nMAssay Description:DPP-IV could hydrolyze Gly-Pro-Aminoluciferin at room temperature to generate Aminoluciferin, which could produce glow type luminescent signals in a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Jiangsu Tasly Diyi Pharmaceutical

US Patent
LigandPNGBDBM408610(US10358449, Compound I-2)
Affinity DataIC50: 2.10nMAssay Description:DPP-IV could hydrolyze Gly-Pro-Aminoluciferin at room temperature to generate Aminoluciferin, which could produce glow type luminescent signals in a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Jiangsu Tasly Diyi Pharmaceutical

US Patent
LigandPNGBDBM408612(US10358449, Compound I-4)
Affinity DataIC50: 4.80nMAssay Description:DPP-IV could hydrolyze Gly-Pro-Aminoluciferin at room temperature to generate Aminoluciferin, which could produce glow type luminescent signals in a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
US Patent