Compile Data Set for Download or QSAR
Report error Found 65 Enz. Inhib. hit(s) with all data for entry = 9163
TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446067(2-chloro-6-fluoro-N-(2-{4-[(3-fluorophenyl)methoxy...)
Affinity DataIC50: 5.95nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446076(N-(2-{4-[(3-fluorophenyl)methoxy]piperidin-1-yl}-2...)
Affinity DataIC50: 11.6nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446071(2-chloro-6-fluoro-N-{2-[4-(3-fluorophenoxy)piperid...)
Affinity DataIC50: 23.6nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446079(N-{2-[4-(4-fluorophenoxy)piperidin-1-yl]-2-(4-meth...)
Affinity DataIC50: 23.9nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446074(2-chloro-N-{2-[4-(3,4-difluorophenoxy)piperidin-1-...)
Affinity DataIC50: 25.8nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446080(N-{2-[4-(3-fluorophenoxy)piperidin-1-yl]-2-(4-meth...)
Affinity DataIC50: 26.4nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446068(2-chloro-6-fluoro-N-(2-{4-[(2-fluorophenyl)methoxy...)
Affinity DataIC50: 28.1nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446083(2-chloro-N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl...)
Affinity DataIC50: 28.9nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446081(N-{2-[4-(2-fluorophenoxy)piperidin-1-yl]-2-(4-meth...)
Affinity DataIC50: 30.2nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446073(2-chloro-N-{2-[4-(3,5-difluorophenoxy)piperidin-1-...)
Affinity DataIC50: 30.6nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446077(N-(2-{4-[(3,5-difluorophenyl)methoxy]piperidin-1-y...)
Affinity DataIC50: 32.9nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446069(2-chloro-N-(2-{4-[(3,5-difluorophenyl)methoxy]pipe...)
Affinity DataIC50: 35.1nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446078(N-(2-{4-[(3,4-difluorophenyl)methoxy]piperidin-1-y...)
Affinity DataIC50: 36.9nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446086(N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl]-2-[4-(4...)
Affinity DataIC50: 39.7nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446084(2-chloro-N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl...)
Affinity DataIC50: 40.7nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446075(N-(2-{4-[(4-fluorophenyl)methoxy]piperidin-1-yl}-2...)
Affinity DataIC50: 42.1nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446072(2-chloro-6-fluoro-N-{2-[4-(2-fluorophenoxy)piperid...)
Affinity DataIC50: 42.9nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446087(N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl]-2-[4-(2...)
Affinity DataIC50: 43.2nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446066(2-chloro-6-fluoro-N-(2-{4-[(4-fluorophenyl)methoxy...)
Affinity DataIC50: 45nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446070(2-chloro-6-fluoro-N-{2-[4-(4-fluorophenoxy)piperid...)
Affinity DataIC50: 51.5nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446085(N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl]-2-{44(3...)
Affinity DataIC50: 56.2nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Human)
Axxam

US Patent
LigandPNGBDBM446082(N-{2-[4-(3,4-difluorophenoxy)piperidin-1-yl]-2-(4-...)
Affinity DataIC50: 57.9nMAssay Description:In order to directly monitor the block of P2X7 channel, an electrophysiological assay was developed and implemented on the QPatch16X automated electr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446087(N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl]-2-[4-(2...)
Affinity DataIC50: 133nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446087(N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl]-2-[4-(2...)
Affinity DataIC50: 133nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446086(N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl]-2-[4-(4...)
Affinity DataIC50: 144nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446086(N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl]-2-[4-(4...)
Affinity DataIC50: 144nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446085(N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl]-2-{44(3...)
Affinity DataIC50: 182nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446082(N-{2-[4-(3,4-difluorophenoxy)piperidin-1-yl]-2-(4-...)
Affinity DataIC50: 201nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446082(N-{2-[4-(3,4-difluorophenoxy)piperidin-1-yl]-2-(4-...)
Affinity DataIC50: 201nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446103(N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl]-2-[4-(3...)
Affinity DataIC50: 216nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446100(N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl]-2-{4-[(...)
Affinity DataIC50: 251nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446095(2-chloro-N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl...)
Affinity DataIC50: 252nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446080(N-{2-[4-(3-fluorophenoxy)piperidin-1-yl]-2-(4-meth...)
Affinity DataIC50: 268nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446080(N-{2-[4-(3-fluorophenoxy)piperidin-1-yl]-2-(4-meth...)
Affinity DataIC50: 268nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446076(N-(2-{4-[(3-fluorophenyl)methoxy]piperidin-1-yl}-2...)
Affinity DataIC50: 288nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446102(N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl]-2-[4-(3...)
Affinity DataIC50: 295nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446101(N-{2-[4-(4-chlorophenoxy)piperidin-1-yl]-2-[4-(dif...)
Affinity DataIC50: 323nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446084(2-chloro-N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl...)
Affinity DataIC50: 329nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446081(N-{2-[4-(2-fluorophenoxy)piperidin-1-yl]-2-(4-meth...)
Affinity DataIC50: 355nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446075(N-(2-{4-[(4-fluorophenyl)methoxy]piperidin-1-yl}-2...)
Affinity DataIC50: 371nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446067(2-chloro-6-fluoro-N-(2-{4-[(3-fluorophenyl)methoxy...)
Affinity DataIC50: 373nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446078(N-(2-{4-[(3,4-difluorophenyl)methoxy]piperidin-1-y...)
Affinity DataIC50: 374nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446074(2-chloro-N-{2-[4-(3,4-difluorophenoxy)piperidin-1-...)
Affinity DataIC50: 380nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446071(2-chloro-6-fluoro-N-{2-[4-(3-fluorophenoxy)piperid...)
Affinity DataIC50: 402nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446077(N-(2-{4-[(3,5-difluorophenyl)methoxy]piperidin-1-y...)
Affinity DataIC50: 432nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446083(2-chloro-N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl...)
Affinity DataIC50: 441nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446099(2-chloro-N-{2-[4-(difluoromethyl)-1,3-thiazol-5-yl...)
Affinity DataIC50: 458nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446069(2-chloro-N-(2-{4-[(3,5-difluorophenyl)methoxy]pipe...)
Affinity DataIC50: 506nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446096(2-chloro-N-{2[4-(difluoromethyl)-1,3-thiazol-5-yl]...)
Affinity DataIC50: 578nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
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TargetP2X purinoceptor 7(Rat)
Axxam

US Patent
LigandPNGBDBM446079(N-{2-[4-(4-fluorophenoxy)piperidin-1-yl]-2-(4-meth...)
Affinity DataIC50: 582nMAssay Description:Ca2+ influx was measured in HEK-293 cells stably transfected with the receptor using Screen Quest Fluo-8 No Wash Calcium Assay Kit (AAt Bioquest ). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details
Go to US Patent

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