Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 9260
TargetAryl hydrocarbon receptor(Human)
Wisconsin Alumni Research Foundation

US Patent
LigandPNGBDBM50049065(CHEMBL3319497 | US9969686, Compound 6 | US10730833...)
Affinity DataEC50:  270nMAssay Description:This assay measures the induction of cytochrome P450-1A1 (CYP1A1), which is a major outcome of AhR activation. Whyte, J. J.; Jung, R. E.; Schmitt, C....More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetAryl hydrocarbon receptor(Human)
Wisconsin Alumni Research Foundation

US Patent
LigandPNGBDBM50049064(CHEMBL3319498 | US9969686, Compound 11a | US107308...)
Affinity DataEC50:  93nMAssay Description:This assay measures the induction of cytochrome P450-1A1 (CYP1A1), which is a major outcome of AhR activation. Whyte, J. J.; Jung, R. E.; Schmitt, C....More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
Go to US Patent

TargetAryl hydrocarbon receptor(Human)
Wisconsin Alumni Research Foundation

US Patent
LigandPNGBDBM50049063(CHEMBL3319499 | US9969686, Compound 11b | US107308...)
Affinity DataEC50:  320nMAssay Description:This assay measures the induction of cytochrome P450-1A1 (CYP1A1), which is a major outcome of AhR activation. Whyte, J. J.; Jung, R. E.; Schmitt, C....More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
Go to US Patent

TargetAryl hydrocarbon receptor(Human)
Wisconsin Alumni Research Foundation

US Patent
LigandPNGBDBM50049062(CHEMBL3319500 | US9969686, Compound 11c | US107308...)
Affinity DataEC50:  230nMAssay Description:This assay measures the induction of cytochrome P450-1A1 (CYP1A1), which is a major outcome of AhR activation. Whyte, J. J.; Jung, R. E.; Schmitt, C....More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
Go to US Patent

TargetAryl hydrocarbon receptor(Human)
Wisconsin Alumni Research Foundation

US Patent
LigandPNGBDBM50049061(CHEMBL3319501 | US9969686, Compound 11d | US107308...)
Affinity DataEC50:  55nMAssay Description:This assay measures the induction of cytochrome P450-1A1 (CYP1A1), which is a major outcome of AhR activation. Whyte, J. J.; Jung, R. E.; Schmitt, C....More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
Go to US Patent

TargetAryl hydrocarbon receptor(Human)
Wisconsin Alumni Research Foundation

US Patent
LigandPNGBDBM50049060(CHEMBL3319502 | US9969686, Compound 6' | US1073083...)
Affinity DataEC50:  215nMAssay Description:This assay measures the induction of cytochrome P450-1A1 (CYP1A1), which is a major outcome of AhR activation. Whyte, J. J.; Jung, R. E.; Schmitt, C....More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
Go to US Patent

TargetAryl hydrocarbon receptor(Human)
Wisconsin Alumni Research Foundation

US Patent
LigandPNGBDBM50049059(CHEMBL3319503 | US9969686, Compound 10a | US107308...)
Affinity DataEC50: >6.70E+3nMAssay Description:This assay measures the induction of cytochrome P450-1A1 (CYP1A1), which is a major outcome of AhR activation. Whyte, J. J.; Jung, R. E.; Schmitt, C....More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
Go to US Patent

TargetAryl hydrocarbon receptor(Human)
Wisconsin Alumni Research Foundation

US Patent
LigandPNGBDBM50049058(CHEMBL3319504 | US9969686, Compound 10c | US107308...)
Affinity DataEC50:  94nMAssay Description:This assay measures the induction of cytochrome P450-1A1 (CYP1A1), which is a major outcome of AhR activation. Whyte, J. J.; Jung, R. E.; Schmitt, C....More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
Go to US Patent

TargetAryl hydrocarbon receptor(Human)
Wisconsin Alumni Research Foundation

US Patent
LigandPNGBDBM50049057(CHEMBL3319505 | US9969686, Compound 10d | US107308...)
Affinity DataEC50:  86nMAssay Description:This assay measures the induction of cytochrome P450-1A1 (CYP1A1), which is a major outcome of AhR activation. Whyte, J. J.; Jung, R. E.; Schmitt, C....More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
Go to US Patent