Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 9329
TargetAdenosine receptor A3(Human)
Palobiofarma

US Patent
LigandPNGBDBM458396(US10744125, Example 5)
Affinity DataKi:  26.3nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
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TargetAdenosine receptor A3(Human)
Palobiofarma

US Patent
LigandPNGBDBM458398(US10744125, Example 14)
Affinity DataKi:  29.2nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
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TargetAdenosine receptor A3(Human)
Palobiofarma

US Patent
LigandPNGBDBM458394(US10744125, Example 4)
Affinity DataKi:  47.6nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
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TargetAdenosine receptor A3(Human)
Palobiofarma

US Patent
LigandPNGBDBM458397(US10744125, Example 6)
Affinity DataKi:  50.3nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
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TargetAdenosine receptor A3(Human)
Palobiofarma

US Patent
LigandPNGBDBM458392(US10744125, Example 3)
Affinity DataKi:  65.5nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
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TargetAdenosine receptor A3(Human)
Palobiofarma

US Patent
LigandPNGBDBM458389(US10744125, Example 1)
Affinity DataKi:  103nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
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TargetAdenosine receptor A1(Human)
Palobiofarma

US Patent
LigandPNGBDBM458398(US10744125, Example 14)
Affinity DataKi: >500nMAssay Description:Adenosine A1 Receptor: Competition assays were carried out by incubation of human recombinant membranes of adenosine receptors from hA1 receptors tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A2a(Human)
Palobiofarma

US Patent
LigandPNGBDBM458398(US10744125, Example 14)
Affinity DataKi: >500nMAssay Description:A2A Adenosine Receptor: Competitive assays were carried out by incubation of membranes from human A2A receptors transfected to HeLa cells, [3H]-ZM241...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A1(Human)
Palobiofarma

US Patent
LigandPNGBDBM458396(US10744125, Example 5)
Affinity DataKi: >500nMAssay Description:Adenosine A1 Receptor: Competition assays were carried out by incubation of human recombinant membranes of adenosine receptors from hA1 receptors tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A2b(Human)
Palobiofarma

US Patent
LigandPNGBDBM458396(US10744125, Example 5)
Affinity DataKi: >500nMAssay Description:A2B Adenosine Receptor: The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A1(Human)
Palobiofarma

US Patent
LigandPNGBDBM458389(US10744125, Example 1)
Affinity DataKi: >500nMAssay Description:Adenosine A1 Receptor: Competition assays were carried out by incubation of human recombinant membranes of adenosine receptors from hA1 receptors tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A2b(Human)
Palobiofarma

US Patent
LigandPNGBDBM458389(US10744125, Example 1)
Affinity DataKi: >500nMAssay Description:A2B Adenosine Receptor: The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A2b(Human)
Palobiofarma

US Patent
LigandPNGBDBM458394(US10744125, Example 4)
Affinity DataKi: >1.00E+3nMAssay Description:A2B Adenosine Receptor: The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A1(Human)
Palobiofarma

US Patent
LigandPNGBDBM458394(US10744125, Example 4)
Affinity DataKi: >1.00E+3nMAssay Description:Adenosine A1 Receptor: Competition assays were carried out by incubation of human recombinant membranes of adenosine receptors from hA1 receptors tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A2a(Human)
Palobiofarma

US Patent
LigandPNGBDBM458394(US10744125, Example 4)
Affinity DataKi: >1.00E+3nMAssay Description:A2A Adenosine Receptor: Competitive assays were carried out by incubation of membranes from human A2A receptors transfected to HeLa cells, [3H]-ZM241...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A2a(Human)
Palobiofarma

US Patent
LigandPNGBDBM458396(US10744125, Example 5)
Affinity DataKi: >1.00E+3nMAssay Description:A2A Adenosine Receptor: Competitive assays were carried out by incubation of membranes from human A2A receptors transfected to HeLa cells, [3H]-ZM241...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A1(Human)
Palobiofarma

US Patent
LigandPNGBDBM458392(US10744125, Example 3)
Affinity DataKi: >1.00E+3nMAssay Description:Adenosine A1 Receptor: Competition assays were carried out by incubation of human recombinant membranes of adenosine receptors from hA1 receptors tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A2b(Human)
Palobiofarma

US Patent
LigandPNGBDBM458392(US10744125, Example 3)
Affinity DataKi: >1.00E+3nMAssay Description:A2B Adenosine Receptor: The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A2a(Human)
Palobiofarma

US Patent
LigandPNGBDBM458392(US10744125, Example 3)
Affinity DataKi: >1.00E+3nMAssay Description:A2A Adenosine Receptor: Competitive assays were carried out by incubation of membranes from human A2A receptors transfected to HeLa cells, [3H]-ZM241...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A2a(Human)
Palobiofarma

US Patent
LigandPNGBDBM458397(US10744125, Example 6)
Affinity DataKi: >1.00E+3nMAssay Description:A2A Adenosine Receptor: Competitive assays were carried out by incubation of membranes from human A2A receptors transfected to HeLa cells, [3H]-ZM241...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A2b(Human)
Palobiofarma

US Patent
LigandPNGBDBM458397(US10744125, Example 6)
Affinity DataKi: >1.00E+3nMAssay Description:A2B Adenosine Receptor: The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A1(Human)
Palobiofarma

US Patent
LigandPNGBDBM458397(US10744125, Example 6)
Affinity DataKi: >1.00E+3nMAssay Description:Adenosine A1 Receptor: Competition assays were carried out by incubation of human recombinant membranes of adenosine receptors from hA1 receptors tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A2b(Human)
Palobiofarma

US Patent
LigandPNGBDBM458398(US10744125, Example 14)
Affinity DataKi: >1.00E+3nMAssay Description:A2B Adenosine Receptor: The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent

TargetAdenosine receptor A2a(Human)
Palobiofarma

US Patent
LigandPNGBDBM458389(US10744125, Example 1)
Affinity DataKi: >1.00E+3nMAssay Description:A2A Adenosine Receptor: Competitive assays were carried out by incubation of membranes from human A2A receptors transfected to HeLa cells, [3H]-ZM241...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
Go to US Patent