Compile Data Set for Download or QSAR
Report error Found 420 Enz. Inhib. hit(s) with all data for entry = 9773
LigandPNGBDBM487269(5-(2,3-Dihydrobenzo[b][1,4]dioxin-6-yl)-7-oxo-N-pr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487268(N-Benzyl-5-(4-chlorophenyl)-7-oxo-4,7-dihydropyraz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487267(N-Benzyl-5-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-N...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487266(2-Amino-5-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-3-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487265(2-Amino-5-(4-chlorophenyl)-3-phenylpyrazolo[1,5-a]...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487264(5-(4-Fluorophenyl)-2-hydroxy-3-(pyridin-2-yl)pyraz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487263(5-(2-Methoxyphenyl)-3-(pyridin-2-yl)pyrazolo[1,5-a...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487262(5-(Benzo[d][1,3]dioxol-5-yl)-3-benzylpyrazolo[1,5-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487261(5-(Benzofuran-5-yl)-2-hydroxy-3-(pyridin-2-yl)pyra...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487260(5-(2,3-Dihydrobenzofuran-5-yl)-2-hydroxy-3-(pyridi...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487259(5-(2,3-Dihydrobenzofuran-5-yl)-2-hydroxy-3-(pyridi...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487258(5-(4-Chlorophenyl)-2-hydroxy-3-(pyridin-3-yl)pyraz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487257(5-(Benzofuran-5-yl)-2-hydroxy-3-phenylpyrazolo[1,5...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487256(5-(3,4-Dichlorophenyl)-3-(pyridin-2-yl)pyrazolo[1,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487255(5-(4-Fluorophenyl)-3-(pyridin-2-yl)pyrazolo[1,5-a]...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487254(5-(4-Chlorophenyl)-2-hydroxy-3-(pyridin-2-yl)pyraz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487286(5-(1H-Benzo[d][1,2,3]triazol-5-yl)-2-hydroxy-3-(py...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487285(2-Amino-5-(1H-benzo[d][1,2,3]triazol-5-yl)-3-(pyri...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487284(2-Amino-5-(4-fluorophenyl)-3-(pyridin-2-yl)pyrazol...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487283(5-(Benzo[d][1,3]dioxol-5-yl)-3-(3-fluoropyridin-2-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487282(2-Amino-5-(4-chloro-2-fluorophenyl)-3-(pyridin-2-y...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487281(5-(Benzo[d][1,3]dioxol-5-yl)-2-ethyl-3-(pyridin-2-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487280(5-(1H-Indazol-5-yl)-3-(pyridin-2-yl)pyrazolo[1,5-a...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487279(US10953012, Example 187 | 2-Amino-5-(1H-indazol-5-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487278(5-(2,2-Difluorobenzo[d][1,3]dioxol-5-yl)-3-(pyridi...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487276(5-(Benzo[d][1,3]dioxol-5-yl)-2-(ethylamino)-3-(pyr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487275(N-(5-(Benzo[d][1,3]dioxol-5-yl)-7-oxo-3-(pyridin-2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487274(2-Amino-5-(4-chlorophenyl)-3-(pyridin-2-yl)pyrazol...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487273(2-Amino-5-(benzo[d][1,3]dioxol-5-yl)-3-(pyridin-2-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487229(US10953012, Example 149 | 5-(Benzofuran-2-yl)-3-(p...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487271(2-Amino-5-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-3-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487270(5-(Benzofuran-5-yl)-2-hydroxy-3-(pyridin-3-yl)pyra...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487309(2-Hydroxy-5-(4-methoxybenzo[d][1,3]dioxol-5-yl)-3-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487308(2-Amino-5-(4-methoxybenzo[d][1,3]dioxol-5-yl)-3-(p...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487306(5-(Benzo[d][1,3]dioxol-5-yl)-2-hydroxy-7-oxo-N-pro...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487305(2-Amino-5-(4-chlorophenyl)-7-oxo-N-propyl-4,7-dihy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487302(2-Amino-5-(3-methyl-1H-indazol-5-yl)-7-oxo-N-propy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487301(2-Amino-5-(1H-benzo[d][1,2,3]triazol-5-yl)-7-oxo-N...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487300(5-(1H-Benzo[d][1,2,3]triazol-5-yl)-3-(4-chlorophen...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487299(2-Amino-5-(1H-benzo[d][1,2,3]triazol-5-yl)-3-(4-ch...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487298(5-(1H-Benzo[d][1,2,3]triazol-5-yl)-7-oxo-N-propyl-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487297(5-(1H-Benzo[d][1,2,3]triazol-5-yl)-3-(pyridin-3-yl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487296(5-(Benzo[d][1,3]dioxol-5-yl)-2-methyl-3-(pyridin-2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487295(N-(5-(1-Methyl-1H-indazol-5-yl)-7-oxo-3-(pyridin-2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487294(5-(1H-benzo[d][1,2,3]triazol-5-yl)-2-ethyl-3-(pyri...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487293(2-Amino-5-(1H-benzo[d][1,2,3]triazol-5-yl)-3-pheny...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487290(2-Amino-5-(1H-indazol-5-yl)-7-oxo-N-propyl-4,7-dih...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487288(2-Amino-5-(1-methyl-1H-indazol-5-yl)-7-oxo-N-propy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 2: Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487320(3-(4-Fluorophenyl)-2-methyl-5-(quinolin-6-yl)pyraz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 3: In the presence of kinase and ATP, the Ulight-peptide is phosphorylated and captured by an anti-phospho-substrate antibody, which brings the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

LigandPNGBDBM487319(5-(2,3-Dihydrobenzo[b][1,4]dioxin-6-yl)-3-(4-metho...)
Affinity DataIC50: 1.00E+4nMAssay Description:Table 3: In the presence of kinase and ATP, the Ulight-peptide is phosphorylated and captured by an anti-phospho-substrate antibody, which brings the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

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