Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 9993
TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506357(methyl ((1S,2R)-2-((S)-1-(1-((1-(4-((1-((E)-4- (di...)
Affinity DataIC50: 1nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506337(methyl ((1S,2R)-2-((S)-(1-((1-(4-((3- acrylamidoph...)
Affinity DataIC50: 2nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506354(methyl ((1S,2R)-2-((S)-cyano(1-((1-(4-((3-((E)-4- ...)
Affinity DataIC50: 2nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506340(methyl ((1S,2R)-2-((S)-1-(1-((1-(4-((1-acryloylaze...)
Affinity DataIC50: 2nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506341(methyl ((1S,2R)-2-((S)-1-(1-((1-(4-((3- acrylamido...)
Affinity DataIC50: 2nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM50511899(CHEMBL4457657 | US11045448, Cpd. No. 67)
Affinity DataIC50: 2nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506342((1S,2R)-2-((S)-(1-((1-(4-((4- acrylamidophenyl)sul...)
Affinity DataIC50: 2nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506346(methyl ((1S,2R)-2-((S)-1-(1-((1-(4-((1-acryloylaze...)
Affinity DataIC50: 2nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM50511900(CHEMBL4454017 | US11045448, Cpd. No. 72)
Affinity DataIC50: 2nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506364(methyl ((1S,2R)-2-((S)-2-(2-ethyl-1H-imidazol-1-yl...)
Affinity DataIC50: 2nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506335((1S,2R)-2-((S)-(1-((1-(4-((3- acrylamidophenyl)sul...)
Affinity DataIC50: 3nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506338(methyl ((1S,2R)-2-((S)-(1-((1-(4-((1-acryloylazeti...)
Affinity DataIC50: 3nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506339(methyl ((1S,2R)-2-((S)-1-(1-((1-(4-((3- acrylamido...)
Affinity DataIC50: 3nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM50511906(CHEMBL4435830 | US11045448, Cpd. No. 57)
Affinity DataIC50: 3nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506365(methyl ((1S,2R)-2-((S)-cyano(3-fluorophenyl)(1-((1...)
Affinity DataIC50: 3nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506352(methyl ((1S,2R)-2-((S)-(1-((1-(4-((4- acrylamidoph...)
Affinity DataIC50: 4nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506353(methyl ((1S,2R)-2-((S)-(1-((1-(4-((3-((E)-but-2- e...)
Affinity DataIC50: 4nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506373(N-((1S,2R)-2-((S)-cyano(1-((1-(4-cyanophenyl)azeti...)
Affinity DataIC50: 4nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506362(methyl ((1S,2R)-2-((S)-cyano(3-fluorophenyl)(1-((1...)
Affinity DataIC50: 4nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506350(methyl ((1S,2R)-2-((S)-cyano(3-fluorophenyl)(1-((1...)
Affinity DataIC50: 4nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506367(2-chloro-N-((1S,2R)-2-((S)-cyano(1-((1-(4- (cyclop...)
Affinity DataIC50: 5nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506347(methyl ((1S,2R)-2-((S)-(1-((1-(4-((1-((E)-but-2-en...)
Affinity DataIC50: 5nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506349(methyl ((1S,2R)-2-((S)-cyano(3-fluorophenyl)(1-((1...)
Affinity DataIC50: 5nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506331((1S,2R)-2-((S)-(1-((1-(4-((1-acryloylazetidin-3- y...)
Affinity DataIC50: 5nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506366(methyl ((1S,2R)-2-((1S)-cyano((2R,6S)-1-((1-(4-((1...)
Affinity DataIC50: 6nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506371(N-((1S,2R)-2-((S)-cyano(1-((1-(4-cyanophenyl)azeti...)
Affinity DataIC50: 7nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506359(methyl ((1S,2R)-2-((S)-cyano(1-(3-(4-((1-((E)-4-(d...)
Affinity DataIC50: 7nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506372(2-chloro-N-((1S,2R)-2-((S)-cyano(1-((1-(4-cyanophe...)
Affinity DataIC50: 9nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506360(methyl ((1S,2R)-2-((S)-cyano(1-((1-(4-((1-((E)-4- ...)
Affinity DataIC50: 9nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506369(methyl ((1S,2R)-2-((1S)-(1-((1-(4-((1-acryloylpipe...)
Affinity DataIC50: 10nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506368(methyl ((1S,2R)-2-((1S)-(1-((1-(4-((1-acryloylpyrr...)
Affinity DataIC50: 11nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506345(methyl ((1S,2R)-2-((S)-(1-((1-(4-((1-acryloylazeti...)
Affinity DataIC50: 24nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506344(methyl ((1S,2R)-2-((S)-(1-((1-(4-((3- acrylamidoph...)
Affinity DataIC50: 42nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506336((1S,2R)-2-((R)-(1-((1-(4-((3- acrylamidophenyl)sul...)
Affinity DataIC50: 300nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506334((1S,2R)-2-((R)-(1-((1-(4-((1-acryloylazetidin-3- y...)
Affinity DataIC50: 374nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506370(N-((1S,2R)-2-((S)-cyano(1-((1-(4-cyanophenyl)azeti...)
Affinity DataIC50: 1.07E+3nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506351(methyl ((1S,2R)-2-((R)-cyano(1-((1-(4-((1-((E)-4- ...)
Affinity DataIC50: 2.00E+3nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506343((1S,2R)-2-((R)-(1-((1-(4-((4- acrylamidophenyl)sul...)
Affinity DataIC50: 2.20E+3nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506355(methyl ((1S,2R)-2-((R)-(4-(2-(4-((1-acryloylazetid...)
Affinity DataIC50: 1.00E+4nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506356(methyl ((1S,2R)-2-((S)-(4-(2-(4-((1-acryloylazetid...)
Affinity DataIC50: 1.00E+4nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandPNGBDBM506361(methyl ((1S,2R)-2-((R)-(1-((1-(4-((3- acrylamidoph...)
Affinity DataIC50: 1.00E+4nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
US Patent