Compile Data Set for Download or QSAR
Report error Found 99 Enz. Inhib. hit(s) with all data for entry = 10427
LigandPNGBDBM534889(1-{5-cyano-6-[(3R)-4- (cyclopropylcarbonyl)-3- met...)
Affinity DataIC50: 5nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534873(1-{5-cyano-6-[(3R)-4- (cyclopropylcarbonyl)-3- met...)
Affinity DataIC50: 5.60nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534875(4-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 8.30nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534891(4-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 9.40nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534894(4-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 9.70nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534897(2-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 10nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534899(2-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 12nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534866(2-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 12nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534888(1-{5-cyano-6-[(3R)-4- (cyclopropylcarbonyl)-3- met...)
Affinity DataIC50: 16nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534879(4-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 19nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534857(3-{2-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiper...)
Affinity DataIC50: 19nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534886(4-(3-amino-1-methyl-1H- pyrazol-4-yl)-2-[(3R)-4- (...)
Affinity DataIC50: 21nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM50537739(CHEMBL4648622 | US11230547, Compound 5-4)
Affinity DataIC50: 21nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534893(4-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 21nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534812(2-(1-methyl-1H-pyrazol-4-yl)-4- {(1S,4R)-5-[3- (me...)
Affinity DataIC50: 27nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534880(4-chloro-2-[(3R)-4- (cyclopropylcarbonyl)-3- methy...)
Affinity DataIC50: 30nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534856(4-{(3R)-3-methyl-4-[3- (methylsulfonyl)phenyl]pipe...)
Affinity DataIC50: 30nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM50537723(CHEMBL4639951 | US11230547, Compound 1-16)
Affinity DataIC50: 31nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534900(4-cyclopropyl-2-[(3R)-4- (cyclopropylcarbonyl)-3- ...)
Affinity DataIC50: 32nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM50537738(CHEMBL4633285 | US11230547, Compound 4-8)
Affinity DataIC50: 32nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534807(2-(1-methyl-1H-pyrazol-4-yl)-4- [(1S,4R)-5-(3-nitr...)
Affinity DataIC50: 38nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534804(4-[(1S,4S)-5-(3-fluorophenyl)- 2,5-diazabicyclo[2....)
Affinity DataIC50: 42nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534890(4-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 49nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534867(2-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 50nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534799(4-[(1R,4S)-5-(3-fluorophenyl)- 2,5-diazabicyclo[2....)
Affinity DataIC50: 51nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM50537721(CHEMBL4646478 | US11230547, Compound 1-17)
Affinity DataIC50: 56nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534884(2-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 58nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534798(4-[(1S,4R)-5-(3-cyanophenyl)- 2,5-diazabicyclo[2.2...)
Affinity DataIC50: 69nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534811(4-[(1S,4R)-5-(3-methoxyphenyl)- 2,5-diazabicyclo[2...)
Affinity DataIC50: 71nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534854(4-[(3R)-3-methyl-4-(3- nitrophenyl)piperazin-1-yl]...)
Affinity DataIC50: 78nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534805(4-{(1S,4R)-5-[3-(2- fluoroethoxy)phenyl]-2,5- diaz...)
Affinity DataIC50: 79nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534878(4-(cyclobutylamino)-6-[(3R)- 4-(cyclopropylcarbony...)
Affinity DataIC50: 80nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534852(4-[(3R)-3-methyl-4-{[(1S,2R)-2- methylcyclopropyl]...)
Affinity DataIC50: 80nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534902(4-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 81nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534887(4-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 83nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534895(4-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 83nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM50537724(CHEMBL4643865 | US11230547, Compound 1-3)
Affinity DataIC50: 86nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534855(4-[(3R)-4-(3-cyanophenyl)-3- melhylpiperazin-1-yl]...)
Affinity DataIC50: 86nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534850(2-(1-methyl-1H-pyrazol-4-yl)-4-[(3R)- 3-methyl-4-(...)
Affinity DataIC50: 87nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534806(2-(1-methyl-1H-pyrazol-4-yl)-4- {(1S,4R)-5-[3-(1H-...)
Affinity DataIC50: 90nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534810(3-{(1R,4S)-5-[5-cyano-2-(1- methyl-1H-pyrazol-4- y...)
Affinity DataIC50: 97nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534818(4-[(1R,4S)-5-(3-fluorophenyl)- 2,5-diazabicyclo[2....)
Affinity DataIC50: 110nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM50537734(CHEMBL4642225 | US11230547, Compound 4-1)
Affinity DataIC50: 110nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534803(2-(1-methyl-1H-pyrazol-4-yl)-4- [(1S,4R)-5-pyridin...)
Affinity DataIC50: 110nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534872(4-amino-6-[(3R)-4- (cyclopropylcarbonyl)-3- methyl...)
Affinity DataIC50: 130nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534808(4-[(1S,4R)-5-(3- cyclopropylphenyl)-2,5- diazabicy...)
Affinity DataIC50: 130nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534876(4-chloro-6-[(3R)-4- (cyclopropylcarbonyl)-3- methy...)
Affinity DataIC50: 140nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534901(4-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 140nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534892(4-[(3R)-4- (cyclopropylcarbonyl)-3- methylpiperazi...)
Affinity DataIC50: 150nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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LigandPNGBDBM534827(4-[(1S,4R)-5-(3-fluoro-2,2- dimethylpropanoyl)-2,5...)
Affinity DataIC50: 160nMAssay Description:This assay was developed and further optimized from a kit produced by Upstate (Millipore catalog #33-047) (Millipore Sigma, Billerica Mass., USA) and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2022
Entry Details
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