Compile Data Set for Download or QSAR
Report error Found 291 Enz. Inhib. hit(s) with all data for entry = 10511
LigandPNGBDBM542862(4-(3-((2-(4-(difluoromethoxy)phenyl)-8-methoxy-2,3...)
Affinity DataIC50: 2nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
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Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542881(3-((2-(6-ethoxypyridin-3-yl)-8-methoxy-2,3-dihydro...)
Affinity DataIC50: 2nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542551(US11274108, Example 1-4 | 3-((2-(4-methoxyphenyl)-...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542814(4-(3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dih...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542815(6-methoxy-3-((8-methoxy-2-(6-methoxypyridin-3-yl)-...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542818(4-(3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dih...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542819(4-(3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dih...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542824(3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dihydr...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542847(3-((2-(6-ethylpyridin-3-yl)-8-methoxy-2,3-dihydrob...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542975(3-(3-methoxy-4-((6-methoxypyridin-3-yl)methoxy)ben...)
Affinity DataIC50: 3nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542518(US11274108, Example 1-2-enant-A | (S)-4-(3-((2-(4-...)
Affinity DataIC50: 4nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542519(US11274108, Example 1-2-enant-B | (S)-4-(3-((2-(4-...)
Affinity DataIC50: 4nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542721(US11274108, Example 1-23 | 4-(3-((2-(6-methoxypyri...)
Affinity DataIC50: 4nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542791((S)-6-(difluoromethyl)-3-((8-methoxy-2-(6-methoxyp...)
Affinity DataIC50: 4nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542813(3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dihydr...)
Affinity DataIC50: 4nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542516(US11274108, Example 1-1 | 4-(1-((2-(4-methoxypheny...)
Affinity DataIC50: 5nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542753(US11274108, Example 1-53 | 3-((8-methoxy-2-(6-meth...)
Affinity DataIC50: 5nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542777(US11274108, Example 1-75 | 6-(1,3-dimethyl-1H-pyra...)
Affinity DataIC50: 5nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542816(3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dihydr...)
Affinity DataIC50: 5nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542820(3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dihydr...)
Affinity DataIC50: 5nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542848(3-((2-(6-ethylpyridin-3-yl)-8-methoxy-2,3-dihydrob...)
Affinity DataIC50: 5nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542974(3-(3-methoxy-4-((6-methoxypyridin-3-yl)methoxy)ben...)
Affinity DataIC50: 5nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542517(US11274108, Example 1-2 | 4-(3-((2-(4-methoxypheny...)
Affinity DataIC50: 6nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542553(US11274108, Example 1-5-enant-A | (S)-4-(3-((2-(6-...)
Affinity DataIC50: 6nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542688(US11274108, Example 1-12 | 4-(3-((2-(4-methoxyphen...)
Affinity DataIC50: 6nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542759(US11274108, Example 1-59 | 4-(3-((8-methoxy-2-(6-m...)
Affinity DataIC50: 6nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542811(6-bromo-3-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,...)
Affinity DataIC50: 6nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542851(4-(3-((8-methoxy-2-(4-methoxyphenyl)-2,3-dihydrobe...)
Affinity DataIC50: 6nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542727(US11274108, Example 1-29 | 4-(3-((8-fluoro-2-(4-(t...)
Affinity DataIC50: 7nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542855(4-(3-((2-(4-(difluoromethoxy)phenyl)-8-methoxy-2,3...)
Affinity DataIC50: 7nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542879(3-((2-(6-ethoxypyridin-3-yl)-8-methoxy-2,3-dihydro...)
Affinity DataIC50: 7nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542944(7-((8-methoxy-2-(6-methoxypyridin-3-yl)-2,3-dihydr...)
Affinity DataIC50: 7nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542761(US11274108, Example 1-60-enant-A | 6-methoxy-3-((8...)
Affinity DataIC50: 8nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542770(US11274108, Example 1-68 | 3-((8-methoxy-2-(6-meth...)
Affinity DataIC50: 8nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542771(US11274108, Example 1-69 | 6-(1H-imidazol-1-yl)-3-...)
Affinity DataIC50: 8nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542831(3-((2-(6-cyclopropylpyridin-3-yl)-8-methoxy-2,3-di...)
Affinity DataIC50: 8nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542852(3-((8-methoxy-2-(4-methoxyphenyl)-2,3-dihydrobenzo...)
Affinity DataIC50: 8nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542754(US11274108, Example 1-54 | 4-(3-((8-methoxy-2-(6-m...)
Affinity DataIC50: 9nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542778(US11274108, Example 1-76 | 6-(6-fluoropyridin-3-yl...)
Affinity DataIC50: 9nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542841(3-((8-methoxy-2-(6-methylpyridin-3-yl)-2,3-dihydro...)
Affinity DataIC50: 9nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542750(US11274108, Example 1-52 | 4-(3-((8-methoxy-2-(6-m...)
Affinity DataIC50: 10nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542860(3-((2-(4-(difluoromethoxy)phenyl)-8-methoxy-2,3-di...)
Affinity DataIC50: 10nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542751(US11274108, Example 1-52-enant-A | 4-(3-((8-methox...)
Affinity DataIC50: 11nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542786(US11274108, Example 1-83-enant-A | azetidin-1-yl(3...)
Affinity DataIC50: 11nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542825(3-((2-(6-cyclopropylpyridin-3-yl)-8-methoxy-2,3-di...)
Affinity DataIC50: 11nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542827(3-((2-(6-cyclopropylpyridin-3-yl)-8-methoxy-2,3-di...)
Affinity DataIC50: 11nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542846(3-((2-(6-ethylpyridin-3-yl)-8-methoxy-2,3-dihydrob...)
Affinity DataIC50: 11nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542737(US11274108, Example 1-39 | 4-(3-((8-fluoro-2-(6-me...)
Affinity DataIC50: 12nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542738(US11274108, Example 1-40 | 3-((8-fluoro-2-(6-metho...)
Affinity DataIC50: 12nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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LigandPNGBDBM542760(US11274108, Example 1-60 | 6-methoxy-3-((8-methoxy...)
Affinity DataIC50: 12nMAssay Description:All assay reaction conditions for IC50 determinations were within the linear range with respect to time and enzyme concentration. In a 384 well polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2022
Entry Details
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