Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 10512
TargetCarbonic anhydrase 2(Human)
Innovative Molecules Gmbg

US Patent
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataIC50: 26nMAssay Description:A protocol for determination of the carbonic anhydrase enzymatic activity at rt using the pH indicator method is described below:1 μL inhibitor ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
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PDB3D3D Structure (crystal)
TargetCarbonic anhydrase 2(Human)
Innovative Molecules Gmbg

US Patent
LigandPNGBDBM50237371(CHEMBL4067954 | US11278534, reference example 87 (...)
Affinity DataIC50: 1.70E+3nMAssay Description:A protocol for determination of the carbonic anhydrase enzymatic activity at rt using the pH indicator method is described below:1 μL inhibitor ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
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TargetCarbonic anhydrase 2(Human)
Innovative Molecules Gmbg

US Patent
LigandPNGBDBM542976( 2-(2′,5′-Difluoro-[1,1′-bipheny...)
Affinity DataIC50: 1.00E+4nMAssay Description:A protocol for determination of the carbonic anhydrase enzymatic activity at rt using the pH indicator method is described below:1 μL inhibitor ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
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TargetCarbonic anhydrase 2(Human)
Innovative Molecules Gmbg

US Patent
LigandPNGBDBM542986((−)-(S)-2-(2′,5′-Difluoro-[1,1&#...)
Affinity DataIC50: 1.00E+4nMAssay Description:A protocol for determination of the carbonic anhydrase enzymatic activity at rt using the pH indicator method is described below:1 μL inhibitor ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
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TargetCarbonic anhydrase 2(Human)
Innovative Molecules Gmbg

US Patent
LigandPNGBDBM542987((+)-(R)-2-(2′,5′-Difluoro-[1,1′-...)
Affinity DataIC50: 1.00E+4nMAssay Description:A protocol for determination of the carbonic anhydrase enzymatic activity at rt using the pH indicator method is described below:1 μL inhibitor ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
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TargetCarbonic anhydrase 2(Human)
Innovative Molecules Gmbg

US Patent
LigandPNGBDBM542988(N-Methyl-N-[4-methyl-5-(methylsulfonimidoyl)thiazo...)
Affinity DataIC50: 1.00E+4nMAssay Description:A protocol for determination of the carbonic anhydrase enzymatic activity at rt using the pH indicator method is described below:1 μL inhibitor ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
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TargetCarbonic anhydrase 2(Human)
Innovative Molecules Gmbg

US Patent
LigandPNGBDBM542989((−)-N-Methyl-N-(4-methyl-5-(S-methylsulfonim...)
Affinity DataIC50: 1.00E+4nMAssay Description:A protocol for determination of the carbonic anhydrase enzymatic activity at rt using the pH indicator method is described below:1 μL inhibitor ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
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TargetCarbonic anhydrase 2(Human)
Innovative Molecules Gmbg

US Patent
LigandPNGBDBM542990((+)-N-Methyl-N-(4-methyl-5-(S-methylsulfonimidoyl)...)
Affinity DataIC50: 1.00E+4nMAssay Description:A protocol for determination of the carbonic anhydrase enzymatic activity at rt using the pH indicator method is described below:1 μL inhibitor ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
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TargetCarbonic anhydrase 2(Human)
Innovative Molecules Gmbg

US Patent
LigandPNGBDBM542991(N-[5-(Cyclopropylsulfonimidoyl)-4-methyl-thiazol-2...)
Affinity DataIC50: 1.00E+4nMAssay Description:A protocol for determination of the carbonic anhydrase enzymatic activity at rt using the pH indicator method is described below:1 μL inhibitor ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
Go to US Patent