Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 10517
LigandPNGBDBM543473(US11279702, Compound 4 | (((6-chloro-5-(2'-hydroxy...)
Affinity DataEC50:  0.550nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
US Patent

LigandPNGBDBM543471(US11279702, Compound 2 | (((6-chloro-5-(2'-hydroxy...)
Affinity DataEC50:  0.970nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
US Patent

LigandPNGBDBM543477(US11279702, Compound 9 | 2-((6-chloro-5-(2'-hydrox...)
Affinity DataEC50:  1.10nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
US Patent

LigandPNGBDBM543470(US11279702, Compound 1 | 2-((6-chloro-5-(2'-hydrox...)
Affinity DataEC50:  1.40nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
US Patent

LigandPNGBDBM543472(US11279702, Compound 3 | ethyl hydrogen (((6-chlor...)
Affinity DataEC50:  2.38nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
US Patent

LigandPNGBDBM543476(US11279702, Compound 8 | 2-((5-(4'-(1H-1,2,4-triaz...)
Affinity DataEC50:  20nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
US Patent

LigandPNGBDBM543475(US11279702, Compound 7 | (S)-2-((6-chloro-5-(4-(3-...)
Affinity DataEC50:  43nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
US Patent

LigandPNGBDBM543469(US11279702, Compound A1)
Affinity DataEC50:  200nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
US Patent

LigandPNGBDBM543474(US11279702, Compound 6 | 2-((6-chloro-5-(4'-(3,3-d...)
Affinity DataEC50:  1.12E+3nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2022
Entry Details
US Patent