Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 10797
TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandPNGBDBM570089(US11427591, Compound 121)
Affinity DataIC50: 7.36nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandPNGBDBM50543781(CHEMBL4632409 | US11427591, Compound 1)
Affinity DataIC50: 9.72nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandPNGBDBM570092(US11427591, Compound 112)
Affinity DataIC50: 11.5nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandPNGBDBM570093(US11427591, Compound 113)
Affinity DataIC50: 12.1nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandPNGBDBM570099(US11427591, Compound 118)
Affinity DataIC50: 13.7nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandPNGBDBM570094(US11427591, Compound 114)
Affinity DataIC50: 14nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandPNGBDBM570086(US11427591, Compound 120)
Affinity DataIC50: 14.6nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandPNGBDBM570084(US11427591, Compound 110)
Affinity DataIC50: 17.3nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandPNGBDBM570096(US11427591, Compound 115)
Affinity DataIC50: 19.3nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandPNGBDBM570090(US11427591, Compound 111)
Affinity DataIC50: 24.5nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandPNGBDBM570097(US11427591, Compound 116)
Affinity DataIC50: 25.8nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandPNGBDBM570098(US11427591, Compound 117)
Affinity DataIC50: 29.1nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandPNGBDBM570085(US11427591, Compound 119)
Affinity DataIC50: 106nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent