Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 10929
TargetWee1-like protein kinase(Human)
Newave Pharmaceutical

US Patent
LigandPNGBDBM579112(2-isopropyl-6-((4-(4-methylpiperazin-1-yl)phenyl)a...)
Affinity DataIC50: 1.5nMAssay Description:In determination of the Weel kinase activity, a synthetic peptide, Poly(Lys,Tyr) Hydrobromide (Lys:Tyr (4:1)) bought from Sigma was used as the subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent

TargetWee1-like protein kinase(Human)
Newave Pharmaceutical

US Patent
LigandPNGBDBM579113(1-(6-(2-fluoropropan-2-yl)pyridin-2-yl)-2-isopropy...)
Affinity DataIC50: 1.5nMAssay Description:In determination of the Weel kinase activity, a synthetic peptide, Poly(Lys,Tyr) Hydrobromide (Lys:Tyr (4:1)) bought from Sigma was used as the subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent

TargetWee1-like protein kinase(Human)
Newave Pharmaceutical

US Patent
LigandPNGBDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)
Affinity DataIC50: 1.5nMAssay Description:In determination of the Weel kinase activity, a synthetic peptide, Poly(Lys,Tyr) Hydrobromide (Lys:Tyr (4:1)) bought from Sigma was used as the subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetWee1-like protein kinase(Human)
Newave Pharmaceutical

US Patent
LigandPNGBDBM579114(1-(6-cyclopropylpyridin-2-yl)-2-isopropyl-6-((4-(4...)
Affinity DataIC50: 1.5nMAssay Description:In determination of the Weel kinase activity, a synthetic peptide, Poly(Lys,Tyr) Hydrobromide (Lys:Tyr (4:1)) bought from Sigma was used as the subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent