Compile Data Set for Download or QSAR
Report error Found 143 Enz. Inhib. hit(s) with all data for entry = 10936
TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579718(US11485711, Compound 146 | 3-ethyl-4-((5-(4-iodoph...)
Affinity DataIC50: 1nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579738(US11485711, Compound 180 | N-(4-((5-(4-(1H-pyrazol...)
Affinity DataIC50: 1nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579704(US11485711, Compound 109 | N-(4-((5-(4-(1H-imidazo...)
Affinity DataIC50: 1nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579709(US11485711, Compound 119 | 4-((5-(5-chlorothiophen...)
Affinity DataIC50: 1nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579739(US11485711, Compound 181 | N-(4-((5-(4-(1H-pyrazol...)
Affinity DataIC50: 2nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579693(US11485711, Compound 81 | 3-ethyl-4-((5-(4- hydrox...)
Affinity DataKd:  3nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579743(US11485711, Compound 187 | N-(4-((5-(4-(1H-pyrazol...)
Affinity DataIC50: 3nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579689(US11485711, Compound 58 | N-(4-((5-(4-hydroxypheny...)
Affinity DataIC50: 3nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579794(US11485711, Compound 265 | 4-((5-(4-(1H-pyrazol-4-...)
Affinity DataIC50: 4nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579686(US11485711, Compound 39 | 4-((5-(4-hydroxyphenyl)-...)
Affinity DataKd:  6nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579714(US11485711, Compound 140 | 4-((5-(1H-indol-3-yl)-1...)
Affinity DataIC50: 6nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579761(US11485711, Compound 205 | 1-(4-(3-((4-hydroxy-2- ...)
Affinity DataIC50: 6nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579764(US11485711, Compound 208 | methyl (4-((5-(4-(1H-py...)
Affinity DataIC50: 7nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579740(US11485711, Compound 182 | 2-(dimethylamino)-N-(4-...)
Affinity DataIC50: 7nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579799(US11485711, Compound 276 | 3-methyl-4-((5-(4-(1-me...)
Affinity DataIC50: 8nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579736(US11485711, Compound 176 | 4-((5-(4-(1H-imidazol-1...)
Affinity DataIC50: 8nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579705(US11485711, Compound 110 | N-(4-((5-(4-(1H-imidazo...)
Affinity DataIC50: 8nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579691(US11485711, Compound 62 | 4-((4-fluoro-5-(4- hydro...)
Affinity DataKd:  8nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579763(US11485711, Compound 207 | 1-(4-((5-(4-(1H-pyrazol...)
Affinity DataIC50: 8nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579687(US11485711, Compound 40 | 4-((5-(4-hydroxyphenyl)-...)
Affinity DataKd:  9nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579765(US11485711, Compound 209 | ethyl (4-((5-(4-(1H-pyr...)
Affinity DataIC50: 9nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579801(US11485711, Compound 278 | 3-methyl-4-((5-(4-(3- (...)
Affinity DataIC50: 9nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579708(US11485711, Compound 117 | 4-((5-(benzo[b]thiophen...)
Affinity DataIC50: 10nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579741(US11485711, Compound 183 | N-(4-((5-(3-fluoro-4- h...)
Affinity DataIC50: 10nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579689(US11485711, Compound 58 | N-(4-((5-(4-hydroxypheny...)
Affinity DataKd:  11nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579800(US11485711, Compound 277 | 4-((5-(4-(3,5-dimethyl-...)
Affinity DataIC50: 11nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579703(US11485711, Compound 86 | N-(4-((5-(4-hydroxy-3- m...)
Affinity DataIC50: 12nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579693(US11485711, Compound 81 | 3-ethyl-4-((5-(4- hydrox...)
Affinity DataIC50: 12nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579696(US11485711, Compound 94 | 2-fluoro-4-((5-(4- hydro...)
Affinity DataKd:  12nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579692(US11485711, Compound 73 | 4-((5-(4-(1H-imidazol-1-...)
Affinity DataKd:  14nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579683(US11485711, Compound 24 | 4-((5-(4-aminophenyl)-1H...)
Affinity DataKd:  14nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579735(US11485711, Compound 175 | 4-((5-(4-(1H-inidazol-1...)
Affinity DataIC50: 15nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579730(US11485711, Compound 170 | N-(4-((5-(4-(1H-imidazo...)
Affinity DataIC50: 15nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579690(US11485711, Compound 59 | N-(4-((5-(4-hydroxypheny...)
Affinity DataKd:  16nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579694(US11485711, Compound 88 | 2-fluoro-4-(3-((4-hydrox...)
Affinity DataKd:  16nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579731(US11485711, Compound 171 | N-(4-((5-(4-(1H-imidazo...)
Affinity DataIC50: 16nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579710(US11485711, Compound 126 | 3-chloro-4-((5-(4- hydr...)
Affinity DataIC50: 17nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579688(US11485711, Compound 49 | 3-fluoro-4-((5-(4- hydro...)
Affinity DataKd:  19nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579798(US11485711, Compound 275 | 2-fluoro-4-((5-(4-hydro...)
Affinity DataIC50: 19nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579797(US11485711, Compound 274 | 4-((5-(4-(1H-pyrazol-1-...)
Affinity DataIC50: 20nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579697(US11485711, Compound 111 | 4-((5-(4-(1H-imidazol-1...)
Affinity DataKd:  20nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579695(US11485711, Compound 89 | 4-((5-(4-hydroxyphenyl)-...)
Affinity DataKd:  21nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579713(US11485711, Compound 139 | N-(4-((5-(4-(1H-pyrazol...)
Affinity DataIC50: 22nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579702(US11485711, Compound 85 | 4-(3-((4-hydroxy-2- meth...)
Affinity DataIC50: 23nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579726(US11485711, Compound 158 | N-(4-((5-(3-fluoro-4- h...)
Affinity DataIC50: 23nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579712(US11485711, Compound 138 | 4-((5-(4-(1H-pyrazol-1-...)
Affinity DataIC50: 23nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579770(US11485711, Compound 215 | 1-(4-(3-((4-hydroxy-2- ...)
Affinity DataIC50: 24nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579804(US11485711, Compound 281 | methyl (4-((5-(4-(1H-py...)
Affinity DataIC50: 25nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579684(US11485711, Compound 29 | N1-(5-(4-chlorophenyl)-1...)
Affinity DataKd:  25nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM579727(US11485711, Compound 160 | 4-(3-((2-ethyl-4- hydro...)
Affinity DataIC50: 26nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

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