Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 10958
TargetKappa-type opioid receptor(Human)
Humanwell Pharmaceutical Us

US Patent
LigandPNGBDBM581036(US11492374, ID 17 | RFCX0139-43)
Affinity DataIC50: 0.157nMAssay Description:The measurement of opioid receptor binding affinity was conducted using a radioligand binding assay on the membranes prepared from HEK293 cells (huma...More data for this Ligand-Target Pair
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Date in BDB:
1/20/2023
Entry Details
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TargetDelta-type opioid receptor(Human)
Humanwell Pharmaceutical Us

US Patent
LigandPNGBDBM581033(US11492374, ID 3)
Affinity DataIC50: 0.158nMAssay Description:The measurement of opioid receptor binding affinity was conducted using a radioligand binding assay on the membranes prepared from HEK293 cells (huma...More data for this Ligand-Target Pair
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Date in BDB:
1/20/2023
Entry Details
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TargetKappa-type opioid receptor(Human)
Humanwell Pharmaceutical Us

US Patent
LigandPNGBDBM581037(US11492374, ID 18 | RFCX0139-45)
Affinity DataIC50: 0.253nMAssay Description:The measurement of opioid receptor binding affinity was conducted using a radioligand binding assay on the membranes prepared from HEK293 cells (huma...More data for this Ligand-Target Pair
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Date in BDB:
1/20/2023
Entry Details
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TargetKappa-type opioid receptor(Human)
Humanwell Pharmaceutical Us

US Patent
LigandPNGBDBM581034(US11492374, ID 13)
Affinity DataIC50: 0.255nMAssay Description:The measurement of opioid receptor binding affinity was conducted using a radioligand binding assay on the membranes prepared from HEK293 cells (huma...More data for this Ligand-Target Pair
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Date in BDB:
1/20/2023
Entry Details
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TargetMu-type opioid receptor(Human)
Humanwell Pharmaceutical Us

US Patent
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataIC50: 0.294nMAssay Description:The measurement of opioid receptor binding affinity was conducted using a radioligand binding assay on the membranes prepared from HEK293 cells (huma...More data for this Ligand-Target Pair
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Date in BDB:
1/20/2023
Entry Details
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TargetKappa-type opioid receptor(Human)
Humanwell Pharmaceutical Us

US Patent
LigandPNGBDBM581035(US11492374, ID 14)
Affinity DataIC50: 0.398nMAssay Description:The measurement of opioid receptor binding affinity was conducted using a radioligand binding assay on the membranes prepared from HEK293 cells (huma...More data for this Ligand-Target Pair
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Date in BDB:
1/20/2023
Entry Details
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TargetKappa-type opioid receptor(Human)
Humanwell Pharmaceutical Us

US Patent
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataIC50: 3.20nMAssay Description:The measurement of opioid receptor binding affinity was conducted using a radioligand binding assay on the membranes prepared from HEK293 cells (huma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2023
Entry Details
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TargetMu-type opioid receptor(Human)
Humanwell Pharmaceutical Us

US Patent
LigandPNGBDBM581034(US11492374, ID 13)
Affinity DataIC50: 4.11E+3nMAssay Description:The measurement of opioid receptor binding affinity was conducted using a radioligand binding assay on the membranes prepared from HEK293 cells (huma...More data for this Ligand-Target Pair
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Date in BDB:
1/20/2023
Entry Details
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TargetMu-type opioid receptor(Human)
Humanwell Pharmaceutical Us

US Patent
LigandPNGBDBM581036(US11492374, ID 17 | RFCX0139-43)
Affinity DataIC50: 5.38E+3nMAssay Description:The measurement of opioid receptor binding affinity was conducted using a radioligand binding assay on the membranes prepared from HEK293 cells (huma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2023
Entry Details
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TargetMu-type opioid receptor(Human)
Humanwell Pharmaceutical Us

US Patent
LigandPNGBDBM581037(US11492374, ID 18 | RFCX0139-45)
Affinity DataIC50: 9.81E+3nMAssay Description:The measurement of opioid receptor binding affinity was conducted using a radioligand binding assay on the membranes prepared from HEK293 cells (huma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2023
Entry Details
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TargetDelta-type opioid receptor(Human)
Humanwell Pharmaceutical Us

US Patent
LigandPNGBDBM581034(US11492374, ID 13)
Affinity DataIC50: 1.00E+4nMAssay Description:The measurement of opioid receptor binding affinity was conducted using a radioligand binding assay on the membranes prepared from HEK293 cells (huma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2023
Entry Details
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TargetMu-type opioid receptor(Human)
Humanwell Pharmaceutical Us

US Patent
LigandPNGBDBM581035(US11492374, ID 14)
Affinity DataIC50: 1.00E+4nMAssay Description:The measurement of opioid receptor binding affinity was conducted using a radioligand binding assay on the membranes prepared from HEK293 cells (huma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2023
Entry Details
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TargetDelta-type opioid receptor(Human)
Humanwell Pharmaceutical Us

US Patent
LigandPNGBDBM581035(US11492374, ID 14)
Affinity DataIC50: 1.00E+4nMAssay Description:The measurement of opioid receptor binding affinity was conducted using a radioligand binding assay on the membranes prepared from HEK293 cells (huma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2023
Entry Details
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TargetDelta-type opioid receptor(Human)
Humanwell Pharmaceutical Us

US Patent
LigandPNGBDBM581036(US11492374, ID 17 | RFCX0139-43)
Affinity DataIC50: 1.00E+4nMAssay Description:The measurement of opioid receptor binding affinity was conducted using a radioligand binding assay on the membranes prepared from HEK293 cells (huma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2023
Entry Details
Go to US Patent

TargetDelta-type opioid receptor(Human)
Humanwell Pharmaceutical Us

US Patent
LigandPNGBDBM581037(US11492374, ID 18 | RFCX0139-45)
Affinity DataIC50: 1.00E+4nMAssay Description:The measurement of opioid receptor binding affinity was conducted using a radioligand binding assay on the membranes prepared from HEK293 cells (huma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2023
Entry Details
Go to US Patent